Serine and cysteine proteases play a central role in digestion, protein degradation and in bioregulation. Their activity may be controlled by activation from inactive proenzyme forms and by inhibition by natural inhibitors. Detailed structural studies have provided a basis for understanding the ...
Serine and cysteine proteases in sul- fur mustard-exposed hairless mouse skin: Enzymatic activity and inhibition profiles. J. Toxicol. Cutan. Ocul. Toxicol. 19, 137-151.Casillas RP, Kam CM, Powers JC. Serine and cysteine proteases in sulfur mustard- exposed hairless mouse skin: enzymatic ...
A novel class of peptide 伪-ketoamides useful for selectively inhibiting serine proteases, selectively inhibiting cysteine proteases, generally inhibiting all serine proteases, and generally inhibiting all cysteine proteases, having the formula M 1 --AA--NH--CHR 2 --CO--CO--NR 3 R 4 , M 1...
A number of cysteine and serine protease inhibitors blocked the intracellular growth and replication of Toxoplasma gondii tachyzoites. Most of these inhibitors caused only minor alterations to parasite morphology irrespective of the effects on the host cells. However, three, cathepsin inhibitor III, TPC...
Results:Collagenaseandserineproteinaseactivitiesindiscsfrom model subgroups wereobviouslyhigherthanthoseofcontrolsubgroups. 结果:造模组动物颈椎间盘中胶原酶和丝氨酸蛋白酶活性明显高于各自的对照组。 dictsearch.appspot.com 5. Tripeptide aldehyde.Reversiblecompetitiveinhibitorofserineandcysteineproteases. ...
Research has confirmed that peptides and larger protein molecules pass through the mucosal barrier of the gastrointestinal tract. Orally administered serine and cysteine proteases of plant and animal origin also reach blood and lymph as intact, high molecular weight and physiologically active protein mole...
First, assays using non-specific protein substrates on purified fecal and body extracts determined that body-associated activity is almost exclusively dependent on cysteine proteases, and specifically on major allergen Der p 1. By contrast, cysteine and serine proteases contributed similarly to the ...
1.Inhibits also some otherserineand cysteine proteases like bromelain, ficin and papain. 也抑制其他的丝氨酸和半胱氨酸蛋 ,如菠萝蛋 、无花果蛋 和木瓜蛋 。 2.Snake venom thrombin-like enzymes belong to the fibrinogenolytic enzyme family and areserineproteases. ...
摘要: (57) [Abstract] The present invention is directed to inhibitors containing a heterocyclic group related and novel benzothiazole serine proteases or cysteine. It is also described how to use it.收藏 引用 批量引用 报错 分享 文库来源 求助全文 Serine protease inhibitors and cysteine-containing ...
SERSociedad de Educación y Rehabilitación(Spanish: Society for Education and Rehabilitation; Puerto Rico) SERSurface Equivalente Radar(French: Radar Cross Section; stealth) SERSchwab Equity Ratings(investing) SERSentence Error Rate(machine translation evaluation) ...