Inhibition of enzyme activity by free fatty acidsdoi:10.1016/S0021-9258(18)94476-5S V PandeJames F Mead
3) inhibition of enzymatic activity 抑制酶活性4) inhibition of enzyme activity 酶活性抑制 例句>> 5) telomrase inhibiting activity 端粒酶抑制活性6) trypsin-inhibitory activity 胰酶抑制活性 1. Serum trypsin-inhibitory activity in seven species of cultured fish; 七种常见养殖鱼血清胰酶抑制活性...
referred to as TOP2A poisons, increases the concentration of covalent enzyme-cleaved DNA complexes and generates DNA strand breaks. The second class is composed by catalytic TOP2 inhibitors, compounds that prevent TOP2 from carrying out its physiological enzymatic activity.18 ...
Concurrently to the cell cycle impairment, bDMC activates a DNA-damage response, which can be responsible for the slower kinetic in re-entering the cell cycle after the release.36 Our present investigations focus on the activity of bDMC as DNA-damaging agent and inhibitor of TOP2A. We high...
It was determined that flavan-3-ols and procyanidins have an inhibitory effect on angiotensin I converting enzyme (ACE) activity, and the effect was dependent on the number of epicatechin units forming the procyanidin. The inhibition by flavan-3-ols and procyanidins was competitive with the two ...
CONSTITUTION:Peroxidase is blended with sodium azide and polyalkylene glycol expressed by formula I (R1, R2, X and Y are hydrogen or lower alkyl; n is integer of >=2) to prepare the peroxidase-containing reagent composition. Inhibition of enzyme activity of peroxidase is prevented by adding ...
Novel 3-chloro-6-nitro-1H-indazole derivatives as promising antileishmanial candidates: synthesis, biological activity, and molecular modelling studies Mohamed Mokhtar Mohamed Abdelahi, Youness El Bakri, Chin-Hung Lai, Karthikeyan Subramani, El Hassane Anouar, Sajjad Ahmad, Mohammed Benchidmi, Joel ...
“flap” covering the dinickel centre of the enzyme, which consequently locks the flap in a specific conformation leading to the loss of catalytic activity. The third category of compounds consists of metal ion chelators, such as EDTA, which can sequester Ni2+, inhibiting the formation of the...
The crude methanolic extract and chloroform, ethyl acetate and n-butanol fractions of Teucrium royleanum were examined as inhibitors of actylcholinesterase, butyrylcholinesterase, lipoxygenase and urease. A significant enzyme inhibition activity (52-83%) was shown by the crude methanolic extract and its...
Inositol requiring enzyme 1 alpha (referred to as IRE1 hereafter, also known as ERN1), an endoplasmic reticulum (ER) resident type I transmembrane protein, is composed of an N-terminal ER luminal domain and a C-terminal cytosolic domain that possesses both kinase and endoribonuclease (RNase) ...