New alpha1-adrenergic receptor antagonist for the treatment of hypertension: role of vascular alpha receptors in the control of peripheral resistance. Am Heart J 1988; 116:160-178.CUBEDDU, L.X. ( 1988 ). New alpha 1-adrenergic receptor antagonists for the treatment of hypertension: role of ...
图1.Dapiprazole hydrochloride化学结构 Dapiprazole hydrochloride基础信息 中文名:盐酸达哌唑;α1-肾上腺素受体拮抗剂;达哌唑; 英文名:Dapiprazole hydrochloride;α1-adrenoreceptor antagonist;alpha1-adrenoreceptor antagonist;Rev-Ey 发布于 2023-04-14 10:24・IP 属地天津 ...
1. Objective To investigate the efficacy and safety of alfuzosin,an alpha-1 adrenoceptor antagonist,on the treatment of neurogenic voiding dysfunction. 目的在神经源性膀胱排空障碍患者中应用α-1肾上腺素能受体阻滞剂阿夫唑嗪,观察其疗效和安全性。6...
Alpha-adrenergic receptor 1a Alpha-adrenergic receptor 1c alpha-adrenergic receptors alpha-adrenoceptor alpha-adrenoceptor antagonist alpha-adrenoceptor antagonist alpha-adrenoceptor blocking drugs Alpha-adrenoreceptor antagonists Alpha-adrenoreceptor antagonists Alpha-agonist Alpha-agonist Alpha-agonist alpha-allocor...
The alpha1 adrenergic receptor antagonist prazosin reduces heroin self-administration in rats with extended access to heroin administration. Pharmacol Biochem Behav 91: 295–302. Grenhoff J, Nisell M, Ferre S, Aston-Jones G, Svensson TH (1993). Noradrenergic modulation of midbrain dopamine cell ...
If an agonist occupies the receptor, a biological process such as enzyme activation, ion influx or efflux across membranes, or production or utilization of energy is then triggered. If an antagonist binds to the receptor, it does not cause a measurable response, but rather blocks the effects ...
MATERIALS AND METHODS: serum levels of interleukin-1 receptor antagonist (IL-1Ra), soluble tumor necrosis factor alpha receptor type I and type II (sTNF-alphaRI and sTNF-alphaRII), and soluble E-selectin (sE-Sel) were followed over time in ten patients with RRMS who were treated with ...
These results suggest that alpha-mangostin is a novel competitive histamine H1 receptor antagonist in smooth muscle cells. 展开 关键词: alpha-mangostin trachea, guinea-pig histamine histamine H-1, receptor antagonist aorta, rabbit DOI: 10.1016/S0014-2999(96)00562-6 ...
Alpha-1 antitrypsin is a multifunctional glycoprotein which provides to human organisms antiinflammatory immunomodulatory, antimicrobial, and tissue repair capacities. IL, Interleukin; IL-1Ra, interleukin-1 receptor antagonist; LB-4, leukotriene B4; TNF, tumor necrosis factor; HIV, human immunodeficiency ...
role is unknown and it may function as an antagonist of the functional receptors because, in transfected cells, it inhibits thetranscriptional activationby TRs (Koenig et al., 1989; Lazar et al., 1989a). However,neuronsexpressing TRα2 are sensitive to T3in vivo(Guadaño-Ferra...