New alpha1-adrenergic receptor antagonist for the treatment of hypertension: role of vascular alpha receptors in the control of peripheral resistance. Am Heart J 1988; 116:160-178.CUBEDDU, L.X. ( 1988 ). New alpha 1-adrenergic receptor antagonists for the treatment of hypertension: role of ...
Facebook Twitter Google Share on Facebook alpha blocker (redirected fromAdrenergic alpha-antagonist) Thesaurus Medical al′pha-block`er n. any of various substances that interfere with the action of the alpha-receptors. al′pha-block`ing,adj. ...
Reduction of human prostate tumor vascularity by the 1-adrenoceptor antagonist terazosin BACKGROUNDWe previously demonstrated that the quinazoline-derived a1-adrenoceptor antagonists doxazosin and terazosin suppress prostate cancer growth via a... K Keledjian,A Borkowski,G Kim,... - 《Prostate》 被引量...
Alpha-1 antitrypsin is a multifunctional glycoprotein which provides to human organisms antiinflammatory immunomodulatory, antimicrobial, and tissue repair capacities. IL, Interleukin; IL-1Ra, interleukin-1 receptor antagonist; LB-4, leukotriene B4; TNF, tumor necrosis factor; HIV, human immunodeficiency ...
A drug combination (CA) formed by ceruletide and alpha-1 antitrypsin showing a predicted value of neuroprotection of 92% was evaluated for their synergic neuroprotective effects in a mouse pre-clinical stroke model. The administration of both drugs in combination was safe and effective in reducing...
This study was designed to assess the effect of alpha-and beta-adrenoceptor antagonist agents on reperfusion ventricular fibrillation and myocardial metabo... FT Thandroyen,MG Worthington,LM Higginson,... - 《Journal of the American College of Cardiology》 被引量: 102发表: 1983年 The effects of...
The pA2 values for antagonist inhibition of alpha-adrenergic receptor-mediated contractile responses were highly correlated (r = 0.995) with the KD values for antagonist inhibition of 125IBE binding in this tissue. The EC50 values for partial agonists were also highly correlated with the KD values...
A comparison of the antagonistic activities of tamsulosin and terazosin against human vascular alpha1-adrenoceptors. Tamsulosin, a selective alpha1A-adrenoceptor antagonist, and terazosin, a non-selective one, are effective for the treatment of urinary disturbance due to ......
Choose the drug which is a H2-receptor antagonist. a) Omeprazole b) Pirenzepine c) Carbenoxolone d) Ranitidine Which of the following drugs has both alfa1-selective and beta-blocking effects? a) Labetalol b) Betaxolol c) Propranolol d) Timolol ...
DISCUSSION When infused into the medial NAc shell, but not the VTA, the a1AR antagonist, terazosin, blunted cocaine- and morphine-induced locomotion and cocaine-induced in- creases in local extracellular DA. The enrichment of these receptors on pre-synaptic glutamatergic, dopaminergic, and GABA...