Procainamide 是一种特异性强效的 DNA 甲基转移酶 1 (DNMT1) 抑制剂。普鲁卡因胺是一种 1A 类抗心律失常药物。Procainamide 具有研究癌症和心律失常的潜力。 ProcainamideChemical Structure CAS No. :51-06-9 *Please selectQuantitybefore adding items. Procainamide 的其他形式现货产品: Procainamide hydrochloride 所...
产品数:86095 上海陶术生物科技有限公司主营产品:生物试剂,实验服务等 第6年 价格:¥电议 型号:T60322原产地:中国大陆更新时间:2025/2/13 11:34:47 产品摘要:Procainamide is a specific and potent DNA methyltransferase 1 ( DNMT1 ) inhibitor. Procainamide is a Class 1A antiarrhythmic agent. Procainamide...
Procainamide is a class 1a antiarrhythmic agent whose primary mechanism is related to its antagonism of cardiac sodium channels delaying phase 0 of the cardiac cycle. Procainamide and its metabolite N -acetyl procainamide also exert potassium efflux channel blocking effects prolonging the QT interval. ...
Procainamide is a class 1a antiarrhythmic that has a mechanism that resembles quinidine by binding to the transmembrane Nat channels and decreasing the number available for depolarization. This creates a delay of Nat entry into the cardiac myocyte during phase 0 of depolarization. As a result, the...
Package insert / product label Generic name: procainamide hydrochloride Dosage form: injection, solution Drug class: Group I antiarrhythmicsMedically reviewed by Drugs.com. Last updated on Feb 24, 2025.On This Page Description Clinical Pharmacology Indications and Usage Contraindications Warnings Precautions...
Procainamide Hydrochloride is the hydrochloride salt form of procainamide, an amide derivative exhibiting class 1A antiarrhythmic property and analog of procaine. Procainamide hydrochloride reversibly binds to and blocks activated (open) voltage-gated sodium channels, thereby blocks the influx of sodium ions...