A DPP-4 inhibitor containing, as an active ingredient, a peptide represented by formula (1): Xe-Pro/Ala/Hyp-Xa-Xb-Xc-Xd (wherein Xe represents an amino acid residue having an isoelectric point of 5.9-6.3; Pro/Al
5.LINONG JI, et al. 55-OR HSK7653, a Novel Ultralong-Acting DPP-4 Inhibitor, as Monotherapy in Patients with Type 2 Diabetes—A Randomized, Double-Blind, Placebo-Controlled Phase III Trial. ADA’s 83rd Scientific Se...
[1]中国医师协会内分泌代谢科医师分会 .DPP-4抑制剂临床应用专家共识.中华内分泌代谢杂志, 2018,34(11) : 899-903 [2]Dianna J Magliano(Co-chair),et al.IDF Diabetes Atlas.2021.[3]Linong Ji,et al.HSK7653, a Novel Ultralong...
5.LINONG JI, et al. 55-OR HSK7653, a Novel Ultralong-Acting DPP-4 Inhibitor, as Monotherapy in Patients with Type 2 Diabetes—A Randomized, Double-Blind, Placebo-Controlled Phase III Trial. ADA’s 83rd Scientific Sessions, 2023. 6.Q Ren, L Ji, L Li, et al. 642 - Hsk7653, a n...
4.Shi D, Chen L, Li G, et al. Clinical Pharmacokinetics. 2024 Jan. 5.LINONG JI, et al. 55-OR HSK7653, a Novel Ultralong-Acting DPP-4 Inhibitor, as Monotherapy in Patients with Type 2 Diabetes—A Randomized, Double-Blind, Placebo-Controlled Phase III Trial. ADA’s 83rd Scientific ...
CAS号1915007-89-4分子量384.35 密度N/A沸点N/A 分子式C21H15F3N2O2熔点N/A MSDSN/A闪点N/A DPP-4抑制剂1用途 DPP-4 inhibitor 1 (compound 5)是有效的、长效的二肽基肽酶-4 (DPP-4) 的抑制剂,有治疗2型糖尿病的潜力,其 KD 值为0.177 nM。
英文名称:dipeptidyl peptidases inhibitor 产品规格:1mL(10mM)|5mg|10mg|50mg Talabostat mesylate是一种可,特异性的dipeptidyl peptidases抑制剂,能够抑制DPP4的活性,IC50值为1nM。 注:本品仅可用于科研实验,严禁用于临床医疗及其他用途! CAS号:150080-09-4 ...
Although either estrogen or the dipeptidyl peptidase-4 (DPP-4) inhibitor, vildagliptin, reduces myocardial damage following cardiac I/R, their effects on the heart in obese-insulin resistant and estrogen deprived conditions remain unknown. Ovariectomized (O) rats (n=36) were divided to receive ...
17. Parmee, E.R., Sinharoy,R., Xu, F., Givand, J.C. and Rosen, L.A.(2012)Discovery and Development Of The DDP-4 Inhibitor Januvia(Sita-Gliptin), in Case Studies in Modern Drug Discovery and Development（eds X. Huang and R.G. Aslanian）,John Wiley&Sons,Inc., Hoboken, NJ, ...
dipeptidyl peptidases inhibitor产品规格:1mL(10mM)|5mg|10mg|50mg发货周期:1～3天产品价格:询价本产品仅可用于科研实验,严禁用于其他非科研用途!Talabostat mesylate是一种可,特异性的dipeptidyl peptidases抑制剂,能够抑制DPP4的活性,IC50值为1nM。注:本品仅可用于科研实验,严禁用于临床医疗及其他用途!