The dopamine receptor agonist drugs could directly stimulate dopamine receptors without actually inducing dopamine synthesis, as is the case with levodopa. The early agonists (bromocrip-tine and pergolide) were ergot derivatives and have been largely replaced by non-ergot medications (eg, pramipexole, ...
A comparison of the first- and second-generation dopamine receptor agonists does not appear to reveal any significant differences in the adverse effect profile of these drugs, which is likely to reflect the fact that they both have D2receptor agonist effects. However, data from tissue culture and...
Functional studies revealed that (−)-43 was one of the highest dopamine D3 receptor selective (EC50, D2 = 114 nM, D3 = 0.26 nM, D2/D3 = 438) agonist in entire series and (−)-45 was nonselective dopamine D3 receptor agonist with high affinity (EC50 D2 = 2.96 nM and D3 ...
IMPORTANCE: Severe impulse control disorders involving pathological gambling, hypersexuality, and compulsive shopping have been reported in association with the use of dopamine receptor agonist drugs in case series and retrospective patient surveys. These agents are used to treat Parkinson disease, restless...
Antipsychotic properties of the partial dopamine agonist (-)-3-(3-hydroxyphenyl)-N-n-propylpiperidine(preclamol) in schizophrenia. Biol Psychiatry 1998;43:2–11. CAS PubMed Google Scholar Wetzel H, Hillert A, Grunder G, Benkert O. Roxindole, a dopamine autoreceptor agonist, in the ...
中文名称:Brexpiprazole (Dopamine Receptor激动剂)英文名称:Brexpiprazole (Dopamine Receptor激动剂) 有效期:一年产品类别:神经科学 Dopamine Signaling 产品编号产品名称产品包装产品价格 SD9563-5mgBrexpiprazole (Dopamine Receptor激动剂)5mg204.00元 化学信息:
Preclinical and clinical studies on the cardiovascular and renal effects of fenoldopam: A DA-1 receptor agonist Recent research in the area of peripheral dopamine (DA) receptors has led to the identification of two distinct subtypes of DA receptors, activation of whi... Mustafa,F.,Lokhandwala ...
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The dopamine receptoragonistbromocriptinelowers IOP in human eyes when administered orally or topically.97,98This effect is blocked by intravenousmetoclopramide, a dopamine2antagonist, suggesting that this agonist is truly acting through dopamine receptors.97A selective dopamine1agonist, feno...
Selective D-2 dopamine receptor agonist 来自 掌桥科研 喜欢 0 阅读量: 15 申请(专利)号: GB19840011483 申请日期: 1984-05-04 公开/公告号: GB2157950A 公开/公告日期: 1985-11-06 申请(专利权)人: * NELSON RESEARCH AND DEVELOPMENT COMPANY 发明人: ALAN S * HORN 被引量: 4 摘要: ...