环苯扎林在2.5 mg至10 mg的剂量范围内表现出线性药代动力学, 并经历肝肠循环。它与血浆蛋白高度结合。每天给药3次后,药物会积聚,在3至4天内达到稳态,血浆浓度约为单次给药后的四倍。 在健康受试者接受10 mg tid(n = 18)的稳态下,血浆峰值浓度为25.9 ng / mL(范围为12.8至46.1 ng / mL), 并且在8...
【英文名】Cyclobenzaprine 【别名】胺苯环庚烯;胺苯庚烯;Flexeril;Novo-Cycloprine;Flexiban;Yurelax 【剂型】环苯扎林片剂:10mg/片。【药理作用】本品为骨骼肌松弛药,在结构上与三环类抗抑郁药相似,主要作用于中枢神经系统的大脑脑干而非脊髓水平,不作用于神经接头,也不直接作用于骨骼肌,主要作用机制是...
10 mg 6202-23-9 ¥312.00 询底价 产品介绍 Cyclobenzaprine (hydrochloride) (Standard) 是 Cyclobenzaprine (hydrochloride) 的分析标准品。本产品用于研究及分析应用。Cyclobenzaprine hydrochloride (MK130 hydrochloride) 是骨骼肌松弛剂,对中枢神经有活性。更多产品详情查看:www.medchemexpress.cn/cyclobenzaprine-hydr...
1) 货号: 03121637; 2) 中文品名: 环苯扎林N-氧化物标准品; 3) 英文品名: Cyclobenzaprine N-oxide; 4) CAS No. 6682-26-4; 5) 分子式、分子量; C20H21NO;291.39 g.mol-1; 6)同位素含量: N/A; 7) 规格: 10 mg, 100 m
给药途径 口服给药 药品规格 10 规格单位 mg/1 市场分类 仿制药 药品申请号 ANDA077563 标签持有者 Jubilant Cadista Pharmaceuticals Inc. 批准日期 2006-04-04 ATC分类 Centrally-mediated Muscle Relaxation [PE], Muscle Relaxant [EPC] 扩展信息 美国上市信息(52) 美国橙皮书信息(50) VIP...
每日剂量不超过60mg,连续服 药不超过2~3 周。 【药物相互作用】1.中枢神经系统抑制药(如催眠药、抗焦虑药、抗抑郁药等) 可增强本品作用,合用时需密切监控或减少本品用量。2.抗胆碱药可增强本品 的抗胆碱能作用。3.与曲马朵合用可增加癫痫发作的危险性。4.本品结构与三...
Cyclobenzaprine Hydrochloride Available forms, composition and doses of Cyclobenzaprine: Tablets; Oral; Cyclobenzaprine Hydrochloride 10 mg Medical categories: Human: Centrally acting skeletal muscle relaxants Skeletal muscle relaxants Indications and usages, anatomical therapeutic chemical and diseases classification...
Adult: 5 mg orally every 8 hours, may increase the dose to 7.5-10 mg orally every 8 hours as needed Under 15 years of age: Safety and efficacy not established Over 15 years of age: 5 mg orally every 8 hours, may increase the dose to 7.5 mg orally every 8 hours as needed ...
5 mg, 7.5 mg, 10 mg oral tablets 15 mg, 30 mg extended-release oral capsules How should I store cyclobenzaprine? Cyclobenzaprine should be stored at room temperature, between 68 F to 77 F (20 C to 25 C). It can be exposed to temperatures between 59 F to 86 F (15 C to 30 C)...
4.僵硬:环苯扎林(cyclobenzaprine)10-50mg或替扎尼定(Tizanidine,商品名凯莱通)4-36mg/d,必要时加用盐酸曲马多. 相关词条 +cyclobenzaprine hydrochloride 1 . 盐酸环苯扎林 ... 盐酸苯甲嗪分析标准品 cyclizine hydrochloride assay standard886 盐酸环苯扎林cyclobenzaprine hydrochloride098 环戊噻嗪 cyclopenthiazide...