Ritanserin, a specific 5HT 2 receptor antagonist has been shown to increase SWS in man. This study explores the effects of a single dose of ritanserin (5 mgr) on the sleep parameters of 10 healthy female subjects aged 25 to 44 years (X=33.2) whose sex and age matched with 10 patients...
在一实施例中,单独选择性5HT-2C受体激动剂的量和一种或一种以上额外医药剂的量在治疗上对于预防和/或治疗所述病况比较不有效,但当组合时,这些化合物协同作用以预防或治疗所述病况。 例如,可与选择性5HT-2C受体激动剂组合使用的适当医药剂包括抗肥胖剂,诸如载脂蛋白B分泌物/微粒体甘油三酯转移蛋白(apo-B/MTP)...
(诸如,从RegeneronPharmaceuticals,Inc.,Tarrytown,NY和Procter & Gamble Company,Cincinnati,OH购得的AxokineTM)、人类豚鼠相关蛋白(AGRP)、增食欲素受体拮抗剂(ghrelin receptorantagonist)、组胺3受体拮抗剂或反向激动剂、神经调节肽U受体激动剂、去甲肾上腺素能减食欲剂(例如,苯丁胺、吗吲哚(mazindol)和其类似物)和...
NEW COMBINATION OF SEROTONIN AGONIST (5HT2) AND ANTAGONIST (5HT6)AS PHARMACEUTICAL FORMULATION The present invention relates to a kind of prevention or the methods of treatment-related disease 5-HT2C receptors and 5-HT6 receptors, are enough to provide the influence for the treatment of including...
摘要: 本发明涉及新化合物(式I);所述化合物起5HT<Sub>2C</Sub>受体调节剂的作用.这些化合物可用于药物组合物,其应用包括治疗肥胖. 展开 收藏 引用 批量引用 报错 分享 全部来源 免费下载 求助全文 掌桥科研 钛学术 (全网免费下载) 钛学术 钛学术 (全网免费下载) 通过文献互助平台发起求助,成功后即可...
, a D1 dopamine receptor antagonist, for 21 days resulted in an increase in D1 dopamine receptors but produced no change in D2 dopamine receptors. During habituation to locomoto... EJ Hess,LJ Albers,H Le,... - 《Journal of Pharmacology & Experimental Therapeutics》 被引量: 208发表: ...
来自 钛学术 喜欢 0 阅读量: 3 发明人: B·史密斯,J·史密斯 展开 摘要: 本发明涉及新化合物(式I);所述化合物起5HT2C受体调节剂的作用.这些化合物可用于药物组合物,其应用包括治疗肥胖. 展开 收藏 引用 批量引用 报错 分享 全部来源 免费下载 求助全文 钛学术 钛学术 (全网免费下载) 钛学术 (...
Antisaccade, Clinical And Motor Executive Functions In Schizophrenia: Effects Of 5Ht2 Antagonist; Cyproheptadinetinnitusprior treatmentsrelaxationacupuncturecognitive-behavioural treatmentEvidence suggests that frontal 5HT2 receptor sensitivity may be increased in schizophrenia, and that they modulate motor responses...
9-[3-(cis-3,5-Dimethyl-1-piperazinyl)propyl]carbazole (rimcazole) has been characterized as a sigma receptor antagonist that binds to the dopamine transpor... SM Husbands,S Izenwasser,T Kopajtic,... - 《Journal of Medicinal Chemistry》 被引量: 129发表: 1999年 Synthesis, Ligand Binding, ...
Dopamine (D2) and serotonin (5HT2) receptor antagonist CAS# 133454-47-4 Catalog No. BCC2516---Order now to get a substantial discount! Product Name & SizePriceStock Iloperidone: 5mg $17 In Stock Iloperidone: 10mg Please Inquire In Stock Iloperidone: 20mg Please Inquire Please Inquire Il...