[16] Sato S, Mizukami K, Asada T. A preliminary open-label studyof 5-HT1A partial agonist tandospirone for behavioural and psychological symptoms associated with dementia[J]. Int JNeuropsychopharmacol, 2007,10(2):281-2...
[22] Miwa H, Nagahara A, Tominaga K, et al. Efficacy of the 5-HT1A agonist tandospirone citrate in improving symptoms of patients with functional dyspepsia: a randomized controlled trial[J]. Am J Gastroenterol, 2009,104(...
Whitaker-Azmitia, 5-HT1A agonist and dexamethasone reversal of para-chloro- amphetamine induced loss of MAP-2 and synaptophysin immuno- reactivity in adult rat brain, Brain Res. 1677 (1995) 181-192.Azmitia EC, Rubinstein VJ, Strafaci JA, Rios JC, Whitaker-Azmitia PM. 1995. 5-HT1A agonist ...
Catalog No.: A11208 5-HT1A agonist BMY 7378 is a 5-HT1A partial agonist and high affinity α1D adrenoceptor antagonist. Skip to the end of the images gallery Skip to the beginning of the images gallery Grouped product items SizePriceStockQty ...
In 1980, buspirone was found to have anxiolytic potential. This finding initiated the development of the azapirones — highly serotonin 5-HT1A agonist
YL0919, a novel antidepressant candidate with dual activity as a 5-HT1A receptor agonist and a selective serotonin reuptake inhibitor,the IC50 values of YL-0919 inhibiting the uptake of 5-HT into rat cerebral cortical synaptosomes and human recombinant c
Aripiprazole, 98%, a human 5-HT1A receptor partial agonist 品牌: J&K 产品编号: 242605 CAS:129722-12-9 分子式: C23H27Cl2N3O2 分子量: 448.40 纯度: 98% 包装库存价格 暂无数据 基本信息 英文别名7-[4-[4-(2,3-Dichlorophenyl)-1-piperazinyl]butoxy]-3,4-dihydro-2(1H)-quinolinone 7-{4-[...
Rats received daily injections of either 50 or 25 ng of the 5-HT1A receptor agonist 8-OH-DPAT or a vehicle solution into the BLA and mutual-reward choices were measured in a rodent prosocial choice task. Compared to vehicle injections, 8-OH-DPAT significantly increased mutual-reward choices ...
In vivo, F 11440 was 4- to 20-fold more potent than flesinoxan, and 30- to 60-fold more potent than buspirone, in exerting 5-HT1A agonist activity at pre- and postsynaptic receptors in rats (measured by, for example, its ability to decrease hippocampal extracellular serotonin (5-HT) ...
[80–83]. Interestingly, signaling to this pathway depends on the 5-HT1A agonist used [82,84,85]. In addition, the 5-HT1A autoreceptor also activates GIRK potassium channels to inhibit neuronal firing [86–89], and inhibits voltage-gated calcium channel activity to reduce calcium entry [90...