A chemical compound of formula (I) wherein R1 to R3 are independently selected from hydrogen and alkyl; R4 to R7 are independently selected from hydrogen, halogen, hydroxy, alkyl, aryl, amino, monoalkylamino, dialkylamino, alkoxy, aryloxy, alkylthio, arylthio, arylsulfoxyl, arylsulfonyl, ...
Der 5-HT2A-Rezeptor The brain serotonin2Areceptor (5-HT2AR) has been implicated in both the pathology of schizophrenia and the therapeutic action of many atypical antipsychoti... R Hurlemann,A Bauer,K Vogeley,... - 《Nervenheilkunde》 被引量: 0发表: 2006年 Sigma-rezeptor-bindungs...
Mehrere Studien weisen darauf hin, dass der Gallensäure-Farnesoid-X-Rezeptor (FXR) Signale übermittelt (z. B. mittels Fibroblasten-Wachstumsfaktor 15/19), die den Triglycerid- und Glukosestoffwechsel beeinflussen. So wurde eine positive Wirkung des FXR-Agonisten Obeticholsäure auf...
7-ARYLSULFONAMID-2,3,4,5-TETRAHYDRO-1H-BENZOiD枚AZEPINE MIT 5-HT6 REZEPTOR AFFINIT脛T ZUR BEHANDLUNG VON ZENTRALNERVENSYSTEMERKRANKUNGEN 7-aryl sulfonamide-2,3,4,5-tetrahydro-1H-BENZOiD枚AZEPINE WITH 5-HT6 RECEPTOR AFFINITY FOR THE TREATMENT OF CENTRAL NERVOUS SYSTEM DISORDERS...
Die Funktionelle Rolle der Palmitilierung des 5-HT 1A Rezeptor In the present study, we verified that the mouse 5-hydroxytryptamine(1A) (5-HT(1A)) receptor is modified by palmitic acid, which is covalently attached to ... E Papoucheva 被引量: 0发表: 2005年 加载更多来源...
Tropisetron; Unclassified drug; Article; Cancer; Cancer chemotherapy; Drug mechanism; Drug structure; Drug synthesis; Nausea; Structure analysis; Vomiting; Animals; Antiemetics; Antineoplastic Agents; Cocaine; Humans; Receptors, Serotonin, 5-HT3; Serotonin Antagonists; Structure-Activity Relationship; Vomit...
BENKYL(IDENE)-LACTAM-DERIVATE, DEREN HERSTELLUNG UND VERWENDUNG ALS SELEKTIVE (ANT)AGONISTEN VON 5-HT1A- UND/ODER 5-HT1D REZEPTOREN compositions thereof, to processes and intermediates for their preparation, and to their medicinal use as selective agonists and antagonists of serotonin 1 (5-HT)...
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Serotonin 5-HT Summary In 1980, buspirone was found to have anxiolytic potential. This finding initiated the development of the azapirones — highly serotonin 5-HT1Aagonists. The balance of evidence suggests that the azapirones act as partial agonists postsynaptically, but as full agonists ...
1-(HETERO)ARYL-4-(KONDENSIERTES THIAZOL-2-YLALKYL)-PIPERAZIN DERIVATE, DEREN HERSTELLUNG UND DEREN VERWENDUNG IN DER BEHANDLUNG VON 5-HT1A-REZEPTOR VERMITT... Aryl and heteroaryl piperazine derivatives of formula (I) wherein, R1 is hydrogen, halogen, trifluoromethyl, C1-C6 alkyl, C1-C6 alko...