Y-27632, Y27632 靶点 (Target) ROCK I/II 通路 (Pathway) Cell Cycle/DNA Damage--ROCK CAS号 (CAS NO.) 146986-50-7 分子式 (Formula) C14H21N3O 分子量 (Molecular Weight) 247.34 外观 (Appearance) 粉末 纯度 (Purity) ≥98% 溶解性 (Solubility) 溶于DMSO 结构式 (...
Y-27632,Y27632 靶点(Target) ROCK I/II 通路(Pathway) Cell Cycle/DNA Damage--ROCK CAS号(CAS NO.) 146986-50-7 分子式(Formula) C14H21N3O 分子量(Molecular Weight) 247.34 外观(Appearance) 粉末 纯度(Purity) ≥98% 溶解性(Solubility)
中文名称:Y 27632 二盐酸盐; 反式-4-[(R)-1-氨基乙基]-N-(4-吡啶基)环己烷甲酰胺二盐酸盐英文名称:Y-27632 dihydrochloride;Y-27632 2HC CAS:129830-38-2有效期:一年 品牌:Chemleader产地:上海 纯度规格:98%+产品类别:信号通路研究 Product Name: Y-27632 dihydrochloride; Y-27632 2HCl ...
口服30 mg/kg的Y-27632可显著降低自发性高血压大鼠、肾性高血压大鼠和醋酸脱氧皮质酮(DOCA)盐性高血压大鼠的血压,并呈剂量依赖性。当Y-27632以0.55 μL / h的速率通过植入泵连续给药11天后,肿瘤细胞(大鼠中表达Val14-RhoA的MM1细胞)的侵袭明显延迟。通过抑制ROCK, Y-27632治疗减弱缺氧诱导的肺循环血管生成和血...
产品代码:MD-0025 Call for Price: 0592-7821662 产品规格 选择产品规格: 2mg (10mM in 624.4╬╝l DMSO) 加入到愿望清单 发送产品给朋友 Product Description Y27632 is a cell-permeable small molecule Rho-associated kinase (ROCK) inhibitor[1]. Y27632 has been found to prevent apoptosis as well as...
Y-27632 is a potent and selective ATP-competitive inhibitor of Rho-associated kinases (ROCK), with Ki values of 0.22 µM and 0.30 µM for ROCK1 and ROCK2, respectively. In vitro kinase assays demonstrate that Y-27632 exhibits a 20-fold greater preference for ROCK when compared to citro...
Y-27632 dihydrochloride 52604ES08 5mg 52604ES10 10mg 52604ES25 25mg 52604ES50 50mg 52604ES60 100mg 产品描述 Y-27632dihydrochloride(又名Y27632 dihydrochloride,Y 27632 dihydrochloride, Y276322HCl)是一种高效、选择性、ATP竞争性ROCK抑制剂,作用于ROCK1 (p160ROCK)(Ki = 140 nM)和ROCK-II (IC50= 80...
Y-27632 是一种 ROCK-I 和 ROCK-II 抑制剂,具有口服有效性、ATP 竞争性。Y-27632 还抑制分离诱导的小鼠前列腺干或祖细胞凋亡。性价比高,品质保障。
Molecular Weight:320.3 g/mol Purity:≥ 98% Pathway:RHO/ROCK Target:ROCK1; ROCK2 Related products Description Catalog # Format Zoledronic Acid, 50 mg 73572 50 mg Zebularine, 10 mg 72902 10 mg Y-27632 (2HCl), 50 mg 72307 1 Kit
Alternative Names: y27632,Y-27632 2HCl,ROCK inhibitor,ROCK1 inhibitor Chemical Name: trans-4-[(1R)-1-Aminoethyl]-N-4-pyridinylcyclohexanecarboxamide dihydrochloride Purity: ≥98% (HPLC) Molecular Weight: 320.26 Loading... Introduction to Tocris View...