英文别名:ROCK Inhibitor|867017-68-3|TC-S 7001|Azaindole 1|Azaindole-1|ROCK-IN-2|6-Chloro-N4-[3,5-difluoro-4-[(3-methyl-1H-pyrrolo[2,3-b]pyridin-4-yl)oxy]phenyl]-2,4-pyrimidinediamine|6-chloro-4-N-[3,5-difluoro-4-[(3-methyl-1H-pyrrolo[2,3-b]pyridin-4-yl)oxy]phenyl] ...
英文别名 ROCK Inhibitor | 867017-68-3 | TC-S 7001 | Azaindole 1 | Azaindole-1 | ROCK-IN-2 | 6-Chloro-N4-[3,5-difluoro-4-[(3-methyl-1H-pyrrolo[2,3-b]pyridin-4-yl)oxy]phenyl]-2,4-pyrimidinediamine | 6-chloro-4-N-[3,5-difluoro-4-[(3-methyl-1H-pyrrolo[2,3-b]pyridin...
Azaindole 1 (ROCK-IN-2, TC-S 7001),又称氮杂吲哚1,是有口服活性、ATP竞争型的ROCK选择性抑制剂,作用于人ROCK1/2的IC50分别为0.6 nM和1.1 nM,在心血管疾病中有作用。Rho-ROCK信号通路在细胞骨架重塑过程中有重要作用,与导致高血压的血管调节改变的病理生理学有关。
📈 影响因子高达17.6,AbMole|TC-S 7001(目录号 M7388;CAS号:867017-68-3)是一款强效且高度选择性的ROCK抑制剂。💊 TC-S 7001对ROCK1和ROCK2的IC50值分别为0.6和1.1 nM,显示出对ROCK的高度抑制作用。同时,它对TRK和FLT3受体的选择性超过200倍,对其他激酶和心血管相关酶和受体的选择性超过900倍。📉...
TC-S 7001 (also known as BAY-549) is a potent and highly selective ROCK inhibitor (IC50 values are 0.6 and 1.1 nM for human ROCK1 and ROCK2, respectively), which exhibits >200-fold selectivity over TRK and FLT3 receptors, and >900-fold selectivity over a panel of other kinases and ca...
生物活性 for TC-S 7001 TC-S 7001 (also known as BAY-549) is a potent and highly selective ROCK inhibitor (IC50 values are 0.6 and 1.1 nM for human ROCK1 and ROCK2, respectively), which exhibits >200-fold selectivity over TRK and FLT3 receptors, and >900-fold selectivity over a ...
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Purity: ≥98% Storage: Store at -20°C CAS No: 867017-68-3 The technical data provided above is for guidance only. For batch specific data refer to the Certificate of Analysis. Tocris products are intended for laboratory research use only, unless stated otherwise. ...