Ro15-4513用途 Ro15-4513 是咪唑并苯二氮酮衍生物,是苯二氮卓受体 (BZR) 的部分反向激动剂。Ro15-4513 是有效的乙醇拮抗剂。Ro15-4513 具有抗焦虑作用。 Ro15-4513名称 英文名ethyl 8-azido-5-methyl-6-oxo-4H-imidazo[1,5-a][1,4]benzodiazepine-3-carboxylate ...
MCE 国际站:Ro15-4513 产品活性:Ro15-4513 是咪唑并苯二氮酮衍生物,是苯二氮卓受体 (BZR) 的部分反向激动剂。Ro15-4513 是有效的乙醇拮抗剂。Ro15-4513 具有抗焦虑作用。 研究领域:Membrane Transporter/Ion Channel | Neuronal Signaling 作用靶点:GABA Receptor In Vitro: Ro15-4513 usually acts as a pa...
RO 15-4513, [7,9-3H]-化学性质 Concentration: 1 mCi/ml Solvent: Ethanol Specific Activity: 20-40 Ci/mmol 安全信息 RO 15-4513, [7,9-3H]-性质、用途与生产工艺 RO 15-4513, [7,9-3H]-上下游产品信息 上游原料 下游产品 RO 15-4513, [7,9-3H]-生产厂家 ...
搜索Ro15-4513 T16775Ro15-4513;化合物 T16775Ro15-4513 ro15-4513 is imidazobenzodiazepinone derivative and is a partial inverse agonist of benzodiazepine receptors. ro15-4513 is an effective ethanol antagonist. 价格:￥电议型号:T16775产地:中国大陆 1共1页 展台...
Basic informationMore Product Name:RO 15-4513, [7,9-3H]- Synonyms:RO 15-4513, [7,9-3H]- CAS: MF:C15H12N6O3T2 MW:330.33 EINECS: Mol File:Mol File Browse by Nationality Suppliers>China suppliers United States (1)All (1) EnquiryRecommend You Select Member Companies ...
The imidazobenzodiazepine, Ro15-4513, has been shown to antagonize some of the behavioral effects of ethanol (ETOH). In rats having relatively little experience in the open field, the actions of ETOH (0.75 g/kg IP), Ro15-4513 (1.25 mg/kg and 2.5 mg/kg, IP), and Ro15-4513 in combi...
RO15-4513 出版社: BOOK ON DEMAND POD 页数: 0 ISBN: 9785511211053 豆瓣评分 目前无人评价 评价: 写笔记 写书评 加入购书单 分享到 推荐 我来说两句 短评 ··· 热门 还没人写过短评呢 我要写书评 RO15-4513的书评 ··· ( 全部0 条 ) 论坛 ··· 在这本书的论坛里发言 + ...
11 C]Ro15-4513 has been introduced as a positron emission tomography radioligand to image the GABA A ±5 receptor subtype thought to be important in learning, memory and addiction. However, the invivo selectivity of the ligand remains unknown and a full assessment of different analysis approaches...
We performed in vitro and in vivo assays of the metabolism of [ 11C]Ro15-4513 over time in the plasma of mice, rats, monkeys and humans, using a radio-HPLC equipped with a sensitive positron detector, in order to compare the metabolic rates of the radiopharmaceutical agent among the differ...
This suggests that attenuation of ethanol-induced motor incoordination was most likely due to the selective antiethanol effect of Ro15–4513 at the dose range used in the present investigation. The antiethanol effect of intracerebellar Ro15–4513 also reaffirmed the well-known belief that the ...