其二,“免疫+”模式的深入探索。免疫+化疗的持续优化,以及免疫+化疗+靶向治疗,包括与靶向VEGFR、FGFR、PDGFR和c-kit等多个靶点的抗血管生成药物或与SCLC特定分子靶向药物联合应用,有望进一步提升ES-SCLC疗效。同时,免疫+放疗具有协同作用,...
此外,肿瘤新生血管生成也是DTC发生与发展的重要因素。多靶点TKI既可以作用于这些信号通路中的关键位点(如RET,VEGFR,PDGFR,c-KIT和BRAF等),阻断信号通路的异常活化抑制肿瘤增殖,也可以作用血管生成通路中的多个位点(如VEGFR,FGFR,PDGFR),抑...
Entrez Gene IDs 5159 (Human); 18596 (Mouse); 24629 (Rat) Alternate Names beta-type platelet-derived growth factor receptor; CD140 antigen-like family member B; CD140b antigen; CD140b; EC 2.7.10; EC 2.7.10.1; JTK12; PDGF R beta; PDGFR; PDGFR1; PDGFRB; PDGF-R-beta; platelet-derived...
PDGF-B PDGF-C PDGF-D PDGF-R PDGF-R-alpha PDGF-R-beta PDGF1 PDGF2 PDGFA PDGFA PDGFA-Associated Protein 1 PDGFB PDGFB PDGFB PDGFC PDGFC PDGFD PDGFD PDGFR PDGFR PDGFR-1 PDGFR-2 PDGFR-alpha PDGFR-beta PDGFR1 PDGFR2 PDGFRA PDGFRA PDGFRA/BCR fusion PDGFRB PDGFRB PDGFRL PDGG PDGI ▼Co...
Sorafenib (Bay 43-9006) 是一种多激酶抑制剂,抑制 Raf-1、B-Raf、VEGFR2、VEGFR3、VEGFR4、PDGFRβ、FLT3、c-Kit 等 (IC50=6/22/90/15/20/20/57/58 nM),具有口服活性。Sorafenib 具有抗肿瘤活性,可以诱导细胞自噬和凋亡,也可以激动铁死亡。
7180 PathScan(R) PDGFR Activity Assay: Phospho-PDGFR, Phospho-SHP2, Phospho-Akt, and Phospho-p44/42 MAPK (Erk1/2) Multiplex Western Detection Kit Antibody Sampler Kit 1 Kit CNY 5,832 9105 Phospho-Bad Antibody Sampler Kit Antibody Sampler Kit 1 Kit CNY 4,200 9369 GSK-3 Antibody Sampler ...
CD140a, PDGFR alpha, PDGFRA Entrez Gene IDs 5156 (Human); 18595 (Mouse) Gene Symbol PDGFRA Additional PDGF R alpha Products All Products for PDGF R alpha PDGF R alpha cDNA Clones PDGF R alpha ELISA Kits PDGF R alpha Lysates PDGF R alpha Pr...
Sorafenib (Bay 43-9006) 是一种多激酶抑制剂,抑制 Raf-1、B-Raf、VEGFR2、VEGFR3、VEGFR4、PDGFRβ、FLT3、c-Kit 等 (IC50=6/22/90/15/20/20/57/58 nM),具有口服活性。Sorafenib 具有抗肿瘤活性,可以诱导细胞自噬和凋亡,也可以激动铁死亡。
Entrez Gene IDs 5156 (Human); 18595 (Mouse) Alternate Names alpha-type platelet-derived growth factor receptor; CD140 antigen-like family member A; CD140a antigen; CD140a; EC 2.7.10; EC 2.7.10.1; MGC74795; PDGF R alpha; PDGFR alpha; PDGFR2; PDGFRA; PDGFRA/BCR fusion; PDGF-R-alpha;...
PDGFR-β (total) Periostin/OSF-2 PF-4/CXCL4 PGRP-S PIINP PR/PGR PRAS40 (total) PRDX-6 Presenilin-1 NTF Procalcitonin proCollagen alpha-1 proCollagen II Progranulin proMMP-10 proMMP-13 Protein C Receptor Proteinase 3 PSGL-1 PSP-D PTEN (total) PYY (active...