本发明提供了一种能够结合至细胞内PRL-1多肽或PRL-3多肽的抗体,其中所述抗体能够结合至与抗体269,抗体223或抗体318结合的表位.这样的抗-PRL抗体能够结合至细胞内PRL-1或PRL-3.它们可以适合被用作抗癌症或癌症转移的治疗剂,或者在临床诊断中来鉴定PRL-3或PRL-1阳性的患者....
每个调节亚基上有两个cAMP结合位点,当胞内的信息分子cAMP的浓度升高时,cAMP即可结合到PKA调节亚基上的cAMP结合位点,催化亚基与调节亚基解离而被激活,生成活性的PKA,其作用是在ATP的存在下磷酸化许多底物蛋白的丝(苏)氨酸残基。 ©2024 Baidu |由 百度智能云...
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or C6-10 aryl; R9a is hydrogen or C1-8 alkyl, not necessarily substituted by hydroxyl; R10a is hydrogen or C1-8 alkyl, not necessarily substituted by hydroxyl; R11 is hydrogen or C1-8 alkyl; R12 is hydrogen or C1-8 alkyl; R13 is hydrogen or C1-8 alkyl; R14 is CF3 or C1-8 a...
C1-8 alkyl optionally substituted with a hydroxyl group, or C6-10 aryl; R9a is hydrogen or C1-8 alkyl optionally substituted with a hydroxyl group; R10a is hydrogen or C1-8 alkyl optionally substituted with a hydroxyl group; R14 is CF3 or C1-8 alkyl.;EFFECT: increased activity of deri...