Sci. 2020, 10, 623 6 of 19 CAuAprpprlp.elS.ncSi.cti2l.0y22,002a,01t,01,l0e6,2a632s3t 11 different scaffolds have been reported as effective DprE1 inh6i6bofiotf1o91r9s, either ctthooavotaptlhteAAAAAiAenmppApppppptpppmppBBBBBlBllllBiBlp...CaC.C.CCC.eCzeeeBeCBelSSeSSSeBaTS....