This transition occurred with an observed rate constant (298 K) of 800 s-1 in the wild-type, and 2500 s-1 in the F87G mutant, suggesting a significant contribution of the phenylalanine side chain to a reaction step rate limiting the actual spin state transition. These findings are ...
SB‐583831 and SB‐583355 are peptidomimetic molecules containing core amino acids (glycine and phenylalanine, respectively), and structurally related to previously described ligands. A telmisartan analog, GSK1820795A, antagonizes the actions of ‐acylamides at GPR132. The synthetic cannabinoid CP‐55940...