N-Arylcyclohexyl-N-acylamines (I) and their isomers and addn. salts are new: n = 0-3; R,R = H; 1-4C alkyl; or one is 2-4C acyl; or NRR = pyrrolidino; piperidino; or morpholino; R,R = H or 1-3C alkyl; R = 1-6C alkyl; 3-6C cycloalkyl; allyl; propargyl; Ph; or ...
Microwave reactions of primary and secondary amines with imidoylbenzotriazoles 6a−w gave diversely substituted amidines 7a−Aa in 76−94% yields. Convenient preparations of a variety of amides 5a−Ab (87−96%) and imidoylbenzo... AR Katritzky,C Cai,SK Singh - 《Journal of Organic Ch...
9Altmetric Metrics Abstract Enantiomerically pure chiral amines and related amide derivatives are privilege motifs in many pharmacologically active molecules. In comparison to the well-established hydroamination, the transition metal-catalysed asymmetric hydrofunctionalization of enamines provides a complementary ...
FAAH located microsomes and catalyzed the hydrolysis of amide bonds between fatty acids and amines. FAAH hydrolyzes not only NAEs including anandamide, but also oleamide, a sleep-inducing lipid (Fig. 11). FAAH could operate in reverse to form anandamide and oleamide, indicating that FAAH is ...
P. L. Use of Chloroalkenylamines for the Synthesis of 1-Azabicyclo[3.3.0]octane and 1-Azabicyclo[4.3.0]nonane Derivatives. J. Chem. Soc., Perkin Trans. 1 1984, 2477-2489.Gesson et al, " ∀-N-Acyliminium Ion—2-Bromoalkene Cyclizations, " Tetrahedron, vol. 49, No. 11. pp. ...
The anodic oxidation pathways of a variety of triphenylamines and other tertiary aromatic amines have been examined. The initial electron-transfer reaction and the identity and stability of the monocation radicals were studied by electro... ET Seo,RF Nelson,JM Fritsch,... - 《Journal of the Am...
摘要: PROBLEM TO BE SOLVED: To obtain a new optically active triacylated binaphthylamine useful for the development of a readily deprotected and easily reutilizable kinetically asymmetric N-acylating agent and useful for the optical resolution of amines using the asymmetric N-acylating agent....
Hydroxyamines N-acyl derivatives having scavenger activity and useful in acute and chronic pathologies associated with peroxidation and inflammation phenomena 申请(专利)号: EP19930121046 申请日: 1993-12-29 专利号: EP0604995A1 公开公告日: 1994-07-06 主分类号: C07D307/81 申请权利人: LIFEGROUP S....
In addition to the peptides and amines secreted by EECs, recent work has indicated other mediators of luminal surveillance in the gut, particularly lipid mediators that appear not to be derived from EECs. For instance, oleoylethanolamide (OEA) is derived from dietary oleate, and has act...
The evidence was accumulated from two dimensional, thin layer chromatography, field desorption mass spectrometry, and accurate mass measurement of the DANS derivatives of the amines. The acetoxy compounds of putrescine and cadaverine have not previously been reported....