While it is true that N-acyl amide are not yet particularly well known throughout scientific communities, we will argue that they are quite well known throughout all of the plant and animal kingdoms in that they are ubiquitous molecules that are formed from simple fatty acids and amines and ...
FAAH located microsomes and catalyzed the hydrolysis of amide bonds between fatty acids and amines. FAAH hydrolyzes not only NAEs including anandamide, but also oleamide, a sleep-inducing lipid (Fig. 11). FAAH could operate in reverse to form anandamide and oleamide, indicating that FAAH is ...
TCFH–NMI: Direct Access to N-Acyl Imidazoliums for Challenging Amide Bond FormationsChallenging couplings of hindered carboxylic acids with non-nucleophilic amines to form amide bonds can be accomplished in high yields, and in many cases... GL Beutner,IS Young,ML Davies,... - 《Organic Letters...
9Altmetric Metrics Abstract Enantiomerically pure chiral amines and related amide derivatives are privilege motifs in many pharmacologically active molecules. In comparison to the well-established hydroamination, the transition metal-catalysed asymmetric hydrofunctionalization of enamines provides a complementary ...
Stable N-acyl-N,N,N-trialkylammonium fluoroborates have been prepared from tertiary amines and acyl halides followed by exchange of anion to fluoroborate w... JV Paukstelis,MG Kim - 《Journal of Organic Chemistry》 被引量: 74发表: 1974年 Peptide Thioester Synthesis via an Auxiliary-Mediated ...
Summary. The preparation of N -acylsulfonamides is described using primary amines, arylsulfonyl chlorides and acyl chlorides. Reaction of primary aryl amin... AR Massah,D Azadi,H Aliyan,... - Monatshefte für Chemie - Chemical Monthly 被引量: 0发表: 2008年 加载更多0关于...
We describe the preparation of new substituted dioxolo[4,5-b]phenothiazines by two slightly different reaction sequences. N-Arylation of [1,3]benzodioxol-5-amine with organolead or organobismuth reagents afforded N-aryl[1,3]benzodioxol-5-amines; subsequent Bernthsen thionation gave rise to phenot...
摘要: Wang resin linked amines were efficiently converted into amides using acylbenzotriazoles. Cleavage of resins gave the desired amides 7Aa–Gf in 30–99% yields with good to excellent purities.DOI: 10.1016/S0960-894X(02)00278-0 年份: 2002 ...
Regioselectivity of the reactions of 1H-1,2,4-triazol-3-amines with 2-acyl-5,5-dimethylcyclohexane-1,3-diones and 2-dimethylaminomethylidene-5,5-dimethylcy... AA Petrov,AN Kasatochkin - 《Russian Journal of Organic Chemistry》 被引量: 3发表: 2013年 Synthesis of 8,9-dihydro[1,2,4]tr...
The evidence was accumulated from two dimensional, thin layer chromatography, field desorption mass spectrometry, and accurate mass measurement of the DANS derivatives of the amines. The acetoxy compounds of putrescine and cadaverine have not previously been reported....