VX-680 (MK-0457, Tozasertib) is a pan-Aurora inhibitor of Aurora A, Aurora B and Aurora C with Kiapp of 0.6 nM, 18 nM and 4.6 nM, respectively. CAS Number:639089-54-6 Purity: >98% Molecular Weight:464.59 Molecular Formula:C23H28N8OS ...
VX-680 (Tozasertib, MK-0457)是一种pan-Aurora抑制剂,对Aurora A作用最强,无细胞试验中Kiapp为0.6 nM,而对Aurora B/Aurora C的作用较弱,对Aurora A选择性比其他55种激酶高100倍。 溶解性:DMSO Solubility: 93 mg/mL (200.17 mM) 体外研究:
VX-680 (MK-0457,Tozasertib)是一种有效的选择性Aurora激酶小分子抑制剂。 温馨提示:产品仅可用于科研实验,不得用于临床诊断或治疗,不得用于食品或药品。 规格 价格 25mg询价 50mg询价 100mg询价 250mg询价 溶解度 In vitroDMSO90 mg/mL (193.71 mM) ...
产品编号 : C14340 产品名称: 陶扎色替 英文名: VX-680(MK-0457,Tozasertib) 别名: Tozasertib,MK 0457 化学名称: N-[4-[4-(4-Methylpiperazin-1-yl)-6-(3-methyl-1H-pyrazol-5-ylamino)pyrimidin-2-sulfanyl]phenyl]- cyclopropanecarboxamide CAS No. : 639089-54-6...
上海玉博生物科技有限公司 主要致力于“Tozasertib (VX-680, MK-0457, VX6) BioVision-1595-25”的生产销售。多年的“Tozasertib (VX-680, MK-0457, VX6) BioVision-1595-25”生产与销售的经验,与各行业新老用户建立了稳定的合作关系,我公司经营的产品名称深受广大用户信
Tozasertib(Synonyms: VX 680; MK-0457)纯度: 99.94% Tozasertib (VX 680; MK-0457) 是Aurora A/B/C 激酶抑制剂,Ki值分别为 0.6,18,4.6 nM。 TozasertibChemical Structure CAS No. :639089-54-6 *Please selectQuantitybefore adding items. ...
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MK-0457 has in vitro activity against cells expressing wild-type or mutated BCR-ABL, including the T315I BCR-ABL mutation. Three patients with T315I abl-mutated chronic myeloid leukemia (CML) or Philadelphia chromosome (Ph)–positive acute lymphocytic leukemia (ALL) have achieved clinical ...
Notably, the MK-0457/vorinostat regimen was highly active against primary CD34+ chronic myelogenous leukemia (CML) cells and Ba/F3 cells bearing various Bcr/Abl mutations (ie, T315I, E255K, and M351T), as well as IM-resistant K562 cells exhibiting Bcr/Abl-independent, Lyn-dependent ...
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