VX-680/MK-0457;陶扎色替;Tozasertib 分子式:C23H28N8OS分子量:464.59 简介:陶扎色替Tozasertib 是一种Aurora-A,Aurora-B,Aurora-C抑制剂,Ki值为 0.6,18,4.6 nM。 别名:MK-0457; VX 680;Tozasertib ;Cyclopropanecarboxamide, N-[4-[[4-(4-methyl-1-piperazinyl)-6-[(5-methyl-1H-pyrazol-3-yl...
VX-680 (MK-0457, Tozasertib) is a pan-Aurora inhibitor of Aurora A, Aurora B and Aurora C with Kiapp of 0.6 nM, 18 nM and 4.6 nM, respectively. CAS Number:639089-54-6 Purity: >98% Molecular Weight:464.59 Molecular Formula:C23H28N8OS ...
VX-680 (MK-0457,Tozasertib)是一种有效的选择性Aurora激酶小分子抑制剂。 温馨提示:产品仅可用于科研实验,不得用于临床诊断或治疗,不得用于食品或药品。 规格 价格 25mg询价 50mg询价 100mg询价 250mg询价 溶解度 In vitroDMSO90 mg/mL (193.71 mM) ...
上海玉博生物科技有限公司 主要致力于“Tozasertib (VX-680, MK-0457, VX6) BioVision-1595-25”的生产销售。多年的“Tozasertib (VX-680, MK-0457, VX6) BioVision-1595-25”生产与销售的经验,与各行业新老用户建立了稳定的合作关系,我公司经营的产品名称深受广大用户信
Tozasertib(Synonyms: VX 680; MK-0457)纯度: 99.94% Tozasertib (VX 680; MK-0457) 是Aurora A/B/C 激酶抑制剂,Ki值分别为 0.6,18,4.6 nM。 TozasertibChemical Structure CAS No. :639089-54-6 *Please selectQuantitybefore adding items. ...
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MK-0457 (VX-680) is a small-molecule aurora kinase (AK) inhibitor with preclinical antileukemia activity. The T315I BCR-ABL mutation mediates resistance to imatinib, nilotinib, and dasatinib. MK-0457 has in vitro activity against cells expressing wild-type or mutated BCR-ABL, including the T31...
Notably, the MK-0457/vorinostat regimen was highly active against primary CD34+ chronic myelogenous leukemia (CML) cells and Ba/F3 cells bearing various Bcr/Abl mutations (ie, T315I, E255K, and M351T), as well as IM-resistant K562 cells exhibiting Bcr/Abl-independent, Lyn-dependent ...
简介内容:MK-0457 is a pan-Aurora kinase inhibitor (Kis: ). It shows selectivity against more than 190 different kinases.详细内容/ContentTozasertibTozasertib,VX 680,MK-0457 美国TargetMol品牌,原装进口,中国现货,所有产品仅用作科学研究,不为任何个人提供产品和服务TozasertibCAS:639089-54-6产品活性:...
本申请涉及猫用零食的领域,具体公开了一种猫条以及该猫条的制备方法,一种猫条,所述猫条包括以下重量份的组分:大豆乳100120份,芝麻粉1525份,肉糜710份,猫薄荷0.30.5份,茶多酚0.0050.02份,肉碱0.30.5份,牛磺酸510份,水2030份,增稠剂24份,碳酸钠0.10.3份和食盐0.20.8份,其中所述大豆乳是大豆采用酵母菌发酵处...