The meta-diamide insecticide acts on insect GABA receptors (GABARs) as an antagonist that causes firing of a neuron. We present here photochromic GABAR ligands azobenzene-meta-diamides (ABMDAs) by incorporating photoswitchable azobenzene with meta-diamides. ABMDAs showed good isomerization efficiency ...
Themeta-diamide insecticide acts on insect GABA receptors (GABARs) as an antagonist that causes firing of a neuron. We present here photochromic GABAR ligands azobenzene-meta-diamides (ABMDAs) by incorporating photoswitchable azobenzene withmeta-diamides.ABMDAsshowed good isomerization efficiency and ...
BACKGROUND Meta-diamides [3-benzamido-N-(4-(perfluoropropan-2-yl)phenyl)benzamides] show high insecticide activity by acting as antagonists to the insect resistance to dieldrin (RDL) gamma-aminobutyric acid (GABA) receptors. In contrast, low-level antagonist activities ofmeta-diamides have been...
Scanning electron microscopy suggested that F17 may deform and rupture Xoo; and (iii) the majority of brominated meta‐diamides were more active than corresponding fluorinated meta‐diamides, which revealed the antibacterial activity of brominated meta‐diamides for the first time. The pr...
Meta-diamide compoundsInsecticidal activityStructure-activity relationshipContentsIn order to discover a novel insecticide, a series of meta-diamide compounds containing n-butyl group were designed and synthesized. Preliminary bioassay data showed that some of the target compounds exhibited good insecticidal ...
Process for sulfonating a diamide of a meta-phenylenediamine, for example, a film forming polyamide of meta-phenylenediamine and isophthaloyl chloride, with a sulfonating agent, for example, sulfur trioxide, which process comprises contacting the diamide and sulfonating agent in the presence of an...