The meta-diamide (m-diamide) insecticide, Broflanilide, was characterized by its high efficiency, low toxicity and lack of cross-resistance with traditional GABA receptors. In accordance with the principles of drug molecular design, easily derivable sulfur with diverse bioactivities...
Novel meta-diamide insecticides [3-benzamido-N-(4-(perfluoropropan-2-yl)phenyl)benzamides] are a distinct class of insect RDL GABA receptor antagonists that have been suggested to act at or near G336 in the M3 region of the Drosophila RDL GABA receptor. Here, we demonstrate the low-level...
www.nature.com/scientificreports OPEN Efficacy of broflanilide (VECTRON T500), a new meta‑diamide insecticide, for indoor residual spraying against pyrethroid‑resistant malaria vectors Corine Ngufor1,2,3*, Renaud Govoetchan1,2,3, Augustin Fongnikin2,3, Estelle Vigninou2...
In this review, we described a novel mode of action for the meta-diamide insecticide, broflanilide. It is suggested that broflanilide is metabolized to desmethyl-broflanilide and that it acts on a novel site in RDL GABARs, that is, at or close to G336 in the M3 region of Drosophil...
which is characterized in that the polyisophthaloyl metaphenylene diamide solution is mixed with a precipitant in a shaping equipment which rotates at certain speed, the polyisophthaloyl metaphenylene diamide solution dissolves out the pulp-shaped fiber in the shearing condition through the precipitant...
META-DIAMIDE COMPOUNDS FOR CONTROLLING INVERTEBRATE PESTSDisclosed are compounds of Formula (1), N-oxides, and salts thereof, wherein Q, X, Y, A1, A2, L, R1, R2, R3, R4, R5, R6a, R6b, R7 and R8 are as defined in the disclosure. Also disclosed are compositions containing the ...
META-DIAMIDE INSECTICIDESDisclosed are compounds of Formula 1, including all geometric and stereoisomers, are as defined in the disclosure. Also disclosed are compositions containing the compounds of Formula 1 and methods for controlling an invertebrate pest comprising contacting the invertebrate pest or ...
Themeta-diamide insecticide acts on insect GABA receptors (GABARs) as an antagonist that causes firing of a neuron. We present here photochromic GABAR ligands azobenzene-meta-diamides (ABMDAs) by incorporating photoswitchable azobenzene withmeta-diamides.ABMDAsshowed good isomerization efficiency and ...
NAKAO T,BANBA S,NOMURA M,et al.Meta-diamide insecticides acting on distinct sites of RDL GABA receptor from those for conventional noncompetitive antagonists[J].Insect Biochem Mol Biol,2013,43(4):366-375.Nakao T, Banba S, Nomura M, Hirase K (2013) Meta-diamide insecticides acting on ...
Broflanilide is a meta-diamide, discovered and named Tenebenal by Mitsui Chemicals Agro, Inc., which has been identified as a candidate insecticide for use in public health products. Methods To evaluate its potential for use in public health, Tenebenal was screened using an array of ...