Miyachi Y, Yoshioka A, Horio T, et al.: Prurigo pigmentosa: a possible mechanism of action of sulfonamides. Dermatologica 172: 82-88, 1986.Miyachi Y, Yoshioka A, Horio T, Imamura S, Niwa Y. Prurigo pigmentosa: a possible mechanism of action of sulfonamides. Dermatologica 1986;172:82-8...
Tipranavir (formerly known as PNU-140690) is the first of a new class of nonpeptide protease inhibitors, the dihydropyrone sulfonamides. Tipranavir was developed and is marketed by Boehringer Ingelheim with the trade name Aptivuss. It was s
Biological activity, design, synthesis and structure activity relationship of some novel derivatives of curcumin containing sulfonamides. Five series of curcumin derivatives with sulfonamides 3a-3e, 4a-4e, 5a-5e, 6a-6e and 7a-7e have been synthesized and evaluated for in vitro antibacterial a... ...
Many strains of Haemophilus influenzae are resistant to erythromycin alone but are found to be susceptible to erythromycin and sulfonamides used in combination. It is important to note that Staphylococci that are resistant to erythromycin may emerge during erythromycin and/or sulfonamide therapy.21 Pseudo...
G01AE10 — Combinations of sulfonamides G01AE — Sulfonamides G01A — ANTIINFECTIVES AND ANTISEPTICS, EXCL. COMBINATIONS WITH CORTICOSTEROIDS G01 — GYNECOLOGICAL ANTIINFECTIVES AND ANTISEPTICS G— GENITO URINARY SYSTEM AND SEX HORMONESS01EC03 — Dorzolamide S01EC — Carbonic anhydrase inhibitors S01...
The sulfonamides are structural analogues of molecules and are similar to biological molecules normally used by the cell target. By using these pharmacological molecules, metabolic pathways of the organism are blocked, causing an inhibition in the production of nitrogen bases and eventually cell death....
Mode of action and quantitative structure–activity relationship of sulfonamides in biological systems of different complexity (enzymes, bacteria, rat, and... Cordes, Mode of action and quantitative structure-activity correlations of tuberculostatic drugs of the isonicotinic acid hydrazide type 1, J. ...
sulfonamides were investigated to inhibit the downstream enzymes of the pathway: the IspF enzyme ofPlasmodium falciparumand, with slightly lower activity, also the homologue fromM. tuberculosis17. However, to the best of our knowledge, no qualified lead compound targeting MEP-pathway enzymes fromM. ...
Leukotriene B4-induced human melanocyte pigmentation and leukotriene C4-induced human melanocyte growth are inhibited by different isoquinolinesulfonamides. J. Invest. Dermatol. 1992, 98, 55–58. [Google Scholar] [CrossRef] Maeda, K.; Naganuma, M. Topical trans-4-aminomethylcyclohexanecarboxylic acid...
(maximum content of 50 mg/kg) and the least residue corresponds to the sulfa antibiotics (maximum content of 1 mg/kg), however, sulfonamides have a stronger effect on the growth of plants [10,11]. Oxytetracycline (OTC) and sulfadiazine (SD) are the most typical representatives of ...