Laduviglusib (CHIR-99021) (GMP) 是 GMP 级别的 Laduviglusib (HY-10182)。GMP 级别的小分子可用做细胞疗法中的辅助试剂。Laduviglusib 是一种有效的,选择性的,具有口服活性的 GSK-3α/β 抑制剂。 MCE 的所有产品仅用作科学研究或药证申报,我们不为任何个人用途提供产品和服务 在干细胞疗法中,化学小分...
8800 nM (IC50) In Vitro CHIR 99021inhibits human GSK-3β with Kivalues of 9.8 nM. CHIR 99021 is a small organic molecule that inhibits GSK3α and GSK3β by competing for their ATP-binding sites.In vitro kinase assays reveal that CHIR 99021 specifically inhibits GSK3β (IC50=~5 nM) an...
构建肾脏类器官 从小鼠肾脏组织中提取细胞,利用微流体技术结合 3D 打印机制作类器官珠,辅以 Noggin (HY-P7086)、R-spondin-1(HY-P7114)、FGF-4 (HY-P7014)、FGF-basic (HY-P7066)、SB-431542 (HY-10431)、Laduviglusib (HY-10182) 培养,7 天后,得到数千个大小、形状和成分具有高度重复性的肾脏类器官...
货号HY-10182应用领域医疗卫生,化工,生物产业,制药 Laduviglusib (CHIR-99021) 是一种有效的,选择性的,具有口服活性的 GSK-3α/β 抑制剂,IC50 为 10 nM 和 6.7 nM。Laduviglusib 对 GSK-3 的选择性比 CDC2,ERK2 和其他蛋白激酶高 500 倍以上。Laduviglusib 还是一种有效的 Wnt/β-catenin 信号通路...
产品活性:Laduviglusib (CHIR-99021) (GMP) 是 GMP 级别的 Laduviglusib (HY-10182)。Laduviglusib 是一种有效的,选择性的,口服活性的 GSK-3α/β 抑制剂。 研究领域:PI3K/Akt/mTOR | Stem Cell/Wnt | Autophagy 作用靶点:GSK-3 | Wnt | β-catenin | Autophagy In Vitro: Laduviglusib (1-10 ...
Laduviglusib (GMP) | MCELaduviglusib (CHIR-99021) (GMP) is <a href=“/Laduviglusib.html“ class=“link-product“ target=“_blank“>Laduviglusib</a> (HY-10182) produced by using GMP guidelines. GMP small molecules works appropriately as an auxiliary reagent for cell th...
Molecules构建肾脏类器官从小鼠肾脏组织中提取细胞,利用微流体技术结合 3D 打印机制作类器官珠,辅以 Noggin(HY-P7086)、R-spondin-1(HY-P7114)、FGF-4(HY-P7014)、FGF-basic(HY-P7066)、SB-431542(HY-10431) 68、、Laduviglusib(HY-10182)培养,7 天后,得到数千个大小、形状和成分具有高度重复性的肾脏类...
SMA42kDaNOX455kDaGAPDH37kDaGAPDH37kDa构建肾脏类器官从小鼠肾脏组织中提取细胞,利用微流体技术结合3D打印机制作类器官珠,辅以Noggin(HY-P7086)、R-spondin-1(HY-P7114)、FGF-4(HY-P7014)、FGF-basic(HY-P7066)、SB-431542(HY-10431)、Laduviglusib(HY-10182)培养,7天后,得到数千个大小、形状和成分具有...
23、wever,it is also important to maintain the balance between the proliferation and differentiation of NSCs as aberrant NSC proliferation can lead to tumorigenesis.Neural Stem CellsCat.No.HY-15036HY-103361HY-10585HY-10182HY-13012HY-10432HY-10587HY-13642HY-B0166HY-15108HY-14649HY-12071HY-1002...
cancer, and bipolar disorder. Phosphorylation of a protein by GSK-3 usually inhibits the activity of its downstream target. GSK-3 is active in a number of central intracellular signaling pathways, including cellular proliferation, migration, inflammation and immune responses,glucose regulation, and ...