Both assay methods showed that the conversion of enalapril to enalaprilat was rapid, and also indicated that there was initial rapid clearance of enalaprilat from the plasma.doi:10.1002/jps.2600750518Peter J. WorlandUniversity of Melbourne, Clinical Pharmacology Unit, Department of Medicine, Austin ...
to yield an activediacidinhibitor,enalaprilat. AllACE inhibitors, exceptlisinopriland captopril, are administered in their prodrug form so as to improve absolute bioavailability.4It was initially thought that prodrug conversion of an ACE inhibitor to an active diacid form would be curtailed in the ...
(Z)-Guggulsterone | Enalapril maleate | Diminazene aceturate | Ramipril | Sinapinic acid | BMS-265246 | Lisinopril | Peimisine | Enalaprilat dihydrate | Perindopril erbumine | Plantainoside D | Alamandine | Benazepril hydrochloride | Omapatrilat | Resorcinolnaphthalein | Fosinopril sodium | Mca-...
(1-7) | Captopril | Enalapril maleate | MLN-4760 | Perindopril erbumine | Benazepril hydrochloride | Phosphoramidon Disodium | Diminazene aceturate | Quinapril hydrochloride | Cilazapril monohydrate | Enalaprilat dihydrate | Fosinopril sodium | Trandolapril | Ramipril | Moexipril hydrochloride | Omap...