Which of the following antiseizure drugs is a prodrug metabolized to phenobarbital? a) Phenytoin b) Primidone c) Felbamate d) Vigabatrin Prodrug: The prodrug is an inactive form of the drug. After administration, it is metabolized to a ...
Plant derived drugs Drugs in pharmacology is a known substance which is used to treat and prevent the diseases. These drugs can be derived from the plants, animals, or can also be synthesised in laboratory. These drugs must be tested on ani...
One special therapeutic category of ethyl ester prodrugs is the angiotensin-converting enzyme (ACE) inhibitors, such as enalapril and perindopril, where one of the carboxylic acid groups is masked as an ethyl ester making the prodrug more lipophilic (Beaumont et al., 2003). Sacubitril (formerly...
Prednisolone was tapered to a dose of 0.2 to 0.3 mg/kg on alternate days for 12 months in both groups. Therapy with calcium carbonate and enalapril was continued. Dose adjustments Trough (12-hour) levels of tacrolimus were measured using microparticle enzyme immunoassay 2 and 12 weeks after ...
Moreover, considering that many ACE inhibitors, including enalapril, trandolapril, and perindopril, are also activated by carboxylesterase, it would be of special interest to study the combination or specificity of the interactions of these prodrugs and the CES genes and their polymorphisms. ...
1.) IV furosemide (Lasix) 2.) Enalapril (Vasotec) 3.) Metoprolol (Lopressor) 4.) IV morphine sulphate (Morp Opioid antagonists can be used if there is excessive sedation or respiratory depression following surgery. Which one is g...
a. Amiodarone b. Milrinone c. Propanolol d. Enalapril Which of the following is a Corticosteroid? A- Beclomethasone B- Formoterol C- Theophylline D- Azelastine Which of the following contains a Beta-Lactam ring? a) Tetracycline b) Macrolides c) Fluoroquinolones d) P...
Enalapril d. Nifedipine Which category of histamine H1 antagonists is noted for the highest local anesthetic effect? a. Alkylamines (propylamines); i.e. Brompheniramine b. Piperidines; i.e. Loratadine, Fexofenadine c. Ethylenediamines; i.e. Su...
a. Cytokine b. Gibberellic acid c. Florigen d. Auxin e. Abscisic acid Tropic Responses: Tropic responses in higher plants occur as a result of the presence of growth hormones. The tropic response involves growth, and a plant may grow towards or away from the stimuli...
Enalapril Which of the following antiseizure drugs may produce teratogenicity? a) Phenytoin b) Valproate c) Topiramate d) All of the above Which of the following medications is a depolarizing neuromuscular blocker? Why would you...