4. Introduction of Fluorine by Halogen Fluorides : 4.2. Fluorination with Chlorine Monofluoridedoi:10.1055/b-003-111685
Among a series of nepenthone derivatives, N-cyclopropylmethyl-nornepenthone (SLL-020ACP, Fig. 3) was found to be a highly selective and potent KOR agonist (Ki = 0.4 nM; μ/κ = 339, δ/κ = 2034) in vitro and could produce KOR-mediated analgesia in vivo [31]. Despite the fact ...
The introduction and preface to this handsome, newly re-issued, three-volume set of Van Gogh's complete letters (which has a design of suns and cornfields gilded across the spines looking very well on dark blue cloth) is completely fascinating.Edmonds, Richard...
Drescher, J, Byne, W (2012) Introduction to the special issue on “The Treatment of Gender Dysphoric/Gender Variant Children and Adolescents”. Journal of Homosexuality 59: pp. 295-300Drescher, J., & Byne, W. (2012). Introduction to the special issue on "The Treatment of Gender ...
In vivo properties of thiol inhibitors of the three vasopeptidases NEP, ACE and ECE are improved by introduction of a 7-azatryptophan in P2¢ position. J Pept Res 2004;63: 99-107.Inguimbert, N.; Poras, H.; Dhotel, H; Beslot, F.; Scalbert, E.; Bennejean, C.; Renard, P.;...