生物活性 INCB054329 (INCB-054329, INCB-54329)是BET抑制剂,对BRD2-BD1, BRD2-BD2, BRD3-BD1, BRD3-BD2, BRD4-BD1, BRD4-BD2, BRDT-BD1和BRDT-BD2的IC50分别为44 nM, 5 nM, 9 nM, 1 nM, 28 nM, 3 nM, 119 nM和63 nM。[1-3] In Vitro 3μM的INCB054329对16种非BET溴区没有显著抑制...