Guanfacine 是一种去甲肾上腺素能 α2A 激动剂,具有口服活性,对α2A 受体亚型具有高度选择性。Guanfacine 具有产生低血压和镇静作用。Guanfacine 可用于研究多种 PFC 认知障碍,包括妥瑞氏综合征和注意力缺陷多动障碍 (ADHD)。 MCE 的所有产品仅用作科学研究或药证申报,我们不为任何个人用途提供产品和服务 ...
Guanfacine is an oral, centrally-acting alpha 2A adrenergic receptor agonist. It is available in two different formulations, Tenex immediate-release tablets, and Intuniv extended-release tablets. Tenex is used alone or in combination with other medications for the treatment ofhypertension(high blood pr...
guanfacine 英汉医学词典 n.胍法新 专业医学词典 胍法辛,氯压脒,胍福新,二氯苯乙酰胍 与"guanfacine"相近的词条 ... guanethidine guanethidine monosulfate guanethidine monosulphate guanethidine sulfate Guanexil guanfacine guanfacine hydrochloride guanfu base A guanfu base B guanfubase A guanfubase B gu...
INN_ID 3999 INCHIKEY INJOMKTZOLKMBF-UHFFFAOYSA-N 别名 N-AMIDINO-2-(2,6-DICHLOROPHENYL)ACETAMIDE;BENZENEACETAMIDE, N-(AMINOIMINOMETHYL)-2,6-DICHLORO-;GUANFACINE [INN];GUANFACINE [MI];ESTULIC;GUANFACINE [WHO-DD];GUANFACINE [VANDF] 中文名 胍法新 扩展信息 VIP...
英文名 guanfacine hydrochloride CAS号 29110-48-3 熔点213 °C 分子式 C9H10Cl3N3O 分子量 282.554 精确质量 280.988953 PSA 78.97000 LogP 3.53850 外观性状 white 储存条件 保持贮藏器密封、储存在阴凉、干燥的地方,确保工作间有良好的通风或排气装置 稳定性 如果遵照规格使用和储存则不会分解,未有已知危险反应...
Guanfacine的适应症 动脉高血压。 禁忌用于胍法辛 超敏反应,低血压,AV阻断II和III度,最近的心肌梗死,心动过缓,抑郁症,伴随使用三环抗抑郁药。 有限制 违反传导,冠状动脉功能不全,脑动脉粥样硬化,历史抑郁,闭塞性外周动脉疾病,窦性心动过缓,慢性肝功能不全,年龄18岁(缺失的疗效和安全性数据)。
Generally reserved as a last-line treatment option because of guanfacine's ability to cause substantial adverse CNS effects, especially in geriatric patients.Has been used in conjunction with diuretics (e.g., thiazides), producing a greater reduction in BP than is obtained with either drug alone...
The meaning of GUANFACINE is a drug that is an alpha-adrenergic agonist taken orally in the form of its hydrochloride C9H9Cl2N3O·HCl especially to treat hypertension and attention deficit hyperactivity disorder. How to use guanfacine in a sentence.
原料品名 Guanfacine 原料中文名称 胍法辛 中文别名 胍法辛;氯苯乙胍;氯苄酰胺;氯酰胍;胍法新-13C-15N3;N-脒基-2-(2,6-二氯苯基)乙酰胺;胍法辛溶液,101PPM;胍甲霜灵杂质 化学名称 N-(diaminomethylidene)-2-(2,6-dichlorophenyl)acetamide 分子式 C9H9Cl2N3O 分子量 246.096 CAS号 29110-...
guanFACINE General General General **BEERS Drug** Pronunciation: gwahn-fa-seen To hear audio pronunciation of this topic, purchase a subscription or log in. Trade Name(s) Intuniv Intuniv XR Tenex Ther. Class. antihypertensives agents for attention deficit hyperactivity disorder (ADHD) Pharm. Cla...