IC50 & Target:PRMT5 CDK4 CDK6 热销产品:mTRP-2 (180-188)|Diminazene (aceturate)|ReAsH-EDT2|Agomelatine|Tebipenem|alpha-Cyperone|IFN-alpha 2/IFNA2, Mouse (His)|Aldosterone-d7|Alofanib|Lipoic acid Trending products:Recombinant Proteins|Bioactive Screening Libraries|Natural Products|Fluorescent Dye|...
GSK3326595 (EPZ015938) 是一种选择性可逆的蛋白精氨酸甲基转移酶 5 抑制剂,IC50为6.2 nM,具有广谱的抗增殖活性。 规格价格库存数量 1 mg ¥ 186 现货 5 mg ¥ 413 现货 10 mg ¥ 579 现货 25 mg ¥ 1,180 现货 50 mg ¥ 1,980 现货 100 mg ¥ 3,730 现货 200 mg ¥ 5...
IC50 & Target:PRMT5 CDK4 CDK6 热销产品:mTRP-2 (180-188) | Diminazene (aceturate) | ReAsH-EDT2 | Agomelatine | Tebipenem | alpha-Cyperone | IFN-alpha 2/IFNA2, Mouse (His) | Aldosterone-d7 | Alofanib | Lipoic acid Trending products:Recombinant Proteins | Bioactive Screening Libraries ...
CHIR-99021是一种GSK-3α/β抑制剂,IC50为10nM/6.7nM。 注:本品仅可用于科研实验,严禁用于临床医疗及其他用途! CAS号:252917-06-9 别名:CT99021 纯度:99.92% 分子式:C₂₂H₁₈Cl₂N₈ 分子量:465.34 结构式: 储存条件:-20℃,有效期2年,溶入溶剂后-20℃请尽量在一个月内使用。 名称:PARP...
IC50 & Target:PRMT5 CDK4 CDK6 热销产品:mTRP-2 (180-188)|Diminazene (aceturate)|ReAsH-EDT2|Agomelatine|Tebipenem|alpha-Cyperone|IFN-alpha 2/IFNA2, Mouse (His)|Aldosterone-d7|Alofanib|Lipoic acid Trending products:Recombinant Proteins|Bioactive Screening Libraries|Natural Products|Fluorescent Dye|...
GSK3326595 (1616395-22-3) is a potent (IC50?= 6.2nM), selective (>4000-fold over 20 other methyltransferases), SAM uncompetitive, peptide competitive inhibitor of PRMT5.1?PRMT5 inhibition activated the p53 pathway?via?induction of alternative splicing of MDM4 leading to a potent anti-proliferati...
GSK3326595 is a potent, selective, reversible inhibitor of protein arginine methyltransferase 5 (PRMT5) with an IC50 of 6.2 nM. ChemeGen 作为优秀的抑制剂、激动剂及新型生命科学试剂的供应商,致力于为广大科研、商业实验室的科学研究者提供高品质的产品与技术服务,不断促进生命科学领域的新技术发展。
GSK3326595是一种* 的,选择性的,可逆的蛋白精氨酸甲基转移酶5 ((PRMT5)) *,具有广泛的抗增殖活性。 Description GSK3326595 is a potent, selective, reversible inhibitor ofprotein arginine methyltransferase 5 (PRMT5)with anIC50of 6.2 nM. IC50& Target ...
IC50: 6.2 nM (PRMT5)[1] 体外研究GSK3326595(EPZ015938)已进入临床试验,用于治疗实体瘤和非霍奇金淋巴瘤[1]。 参考文献 [1].WO 2016022605 A1 GSK3326595物理化学性质 密度1.3±0.1 g/cm3 沸点760.3±60.0 °C at 760 mmHg 分子式C24H32N6O3
GSK3326595 (EPZ015938) is a potent, selective, reversible inhibitor ofprotein arginine methyltransferase 5 (PRMT5)with anIC50of 6.2 nM[1]. IC50& Target IC50: 6.2 nM (PRMT5)[1] 体外研究 (In Vitro) GSK3326595 (EPZ015938), has entered clinical trials for the treatment of solid tumors and...