Trastuzumab deruxtecan(T-DXd, DS-8201)是由曲妥珠单抗、酶切肽连接体和新型DNA拓扑异构酶I抑制剂德鲁替康组成的靶向HER2的抗体偶联药物。DESTINY-Gastric01研究是一项注册性、前瞻性、多队列的Ⅱ 期临床研究, 评估DS-8201作为HER2阳性胃或胃食管交界癌患者...
[6]Nakada T, Sugihara K, Jikoh T, et al. The latest research and development into the antibody-drug conjugate, [fam-] trastuzumab deruxtecan (DS-8201a), for HER2 cancer therapy. Chem Pharm Bull. 2019;67 (3):173–185. ...
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Chen JR,Yen JH,Lin CC, et al.The effects of Chinese herbs on improving survival and inhibiting anti-ds DNA antibody production in lupus mice. American Journal of Chinese Medicine . 1993Chen JR,et al.The effects of chinese herbs on improving survival and inhibiting anti-dsDNA antibody ...
Learn more about our ImmunoCruz® Antibody Conjugates and Cruz Marker™ MW Standards Promotional描述说明书与实验方案研究信息 脱氧核糖核酸(DNA)是一种核酸,它存储着关于所有已知生物体发育和功能的长期信息。DNA由两个长核苷酸聚合物组成,这两个聚合物由四个碱基组成,即腺嘌呤、胸腺嘧啶、鸟嘌呤和胞嘧啶,所...
ChemicalBook provide Chemical industry users with Anti-ds DNA antibody [35I9 DNA] - BSA and Azide free Boiling point Melting point,Anti-ds DNA antibody [35I9 DNA] - BSA and Azide free Density MSDS Formula Use,If You also need to Anti-ds DNA antibody [35I
Learn more about our ImmunoCruz® Antibody Conjugates and Cruz Marker™ MW Standards Promotional描述说明书与实验方案研究信息 脱氧核糖核酸(DNA)是一种核酸,它存储着关于所有已知生物体发育和功能的长期信息。DNA由两个长核苷酸聚合物组成,这两个聚合物由四个碱基组成,即腺嘌呤、胸腺嘧啶、鸟嘌呤和胞嘧啶,所...
DNA ds & ss antibody [3901] 中文名: 中文别名: CBNumber: CB75727880 分子式: 分子量: 0 MOL File: Mol file 化学性质安全信息用途供应商11 DNA ds & ss antibody [3901]化学性质 安全信息 DNA ds & ss antibody [3901]性质、用途与生产工艺 ...
13.Takegawa, N., et al., Takegawa, N., et al.,DS-8201a, a new HER2-targeting antibody-drug conjugate incorporating a novel DNA topoisomerase I inhibitor, overcomes HER2-positive gastric cancer T-DM1 resistance.Int J Cancer, 2017.141(8): p. 1682-1689. ...
另一方面,DS-8201a(10 mg/mL)可诱导Chk1和组蛋白H2A.X的磷酸化(DNA损伤Marker[19, 20])以及PARP裂解(凋亡Marker[21]),10 mg/mL的抗HER2 Ab在相应时间点都不会引起任何目标蛋白的变化,这些结果表明DS-8201a以与DXd相同的方式诱导DNA损伤和细胞凋亡。因此,D...