It is a potent inhibitor of lysosomal proteinases (enzymes from a special subunit of the cell that break down proteins) and probably one of the most important extracellular inhibitors ofcysteine proteases(it prevents the breakdown of proteins outside the cell by a specific type of protein degrading...
Cysteine protease ATG4A belongs to a member of the autophagin protein family. This protein is also designated as a member of the C-54 family of cysteine proteases. Autophagy is the process by which endogenous proteins and damaged organelles are destroyed intracellularly. Autophagy is postulated to...
信号通路 Proteases 靶点 Cysteine protease - - - - IC50 9nM - - - - 体外研究 E-64迅速抑制半胱氨酸蛋白酶组织蛋白酶B、H 、L和木瓜蛋白酶,而对丝氨酸蛋白酶或金属蛋白酶没有作用。E-64,半胱氨酸蛋白酶的特异性抑制剂,有效阻断体外卵巢癌细胞侵袭。此外,E-64也表现出对贾第鞭毛虫脱囊的体外抗寄生...
产品描述Odanacatib (MK-0822)是一种有效的,选择性的,cathepsin K(人/兔)中性抑制剂,IC50为0.2nM/1nM,对脱靶的cathepsin B、L、S具有高度选择性。Phase 3。 信号通路Proteases 靶点Cathepsin K (human)Cathepsin K (rabbit)--- IC500.2nM1nM---
溶液配制5mg加入1.4ml DMSO,或者每3.57mg加入1ml DMSO,配制成10mM溶液。SF4135-10mM用DMSO配制。 生物信息: 产品描述E-64 is an irreversible and selective cysteine protease inhibitor with IC50 of 9nM for papain. 信号通路Proteases 靶点Cysteine protease--- IC50...
E-64蛋白酶抑制剂 (10mM)价格:￥130.00/瓶产品详情:E-64蛋白酶抑制剂 (10mM)英文名称E-64 solution (10mM)中文名称E-64蛋白酶抑制剂 (10mM)别名trans-Epoxysuccinyl-L-leucylamid... 纯度:99% 包装规格:200ul 用途:E-64 是一种有效的不可逆的半胱氨酸蛋白酶 (cysteine proteases) 抑制剂,抑制 papain 的...
产品描述 Odanacatib (MK-0822)是一种有效的,选择性的,cathepsin K(人/兔)中性抑制剂,IC50为0.2nM/1nM,对脱靶的cathepsin B、L、S具有高度选择性。Phase 3。 信号通路 Proteases 靶点 Cathepsin K (human) Cathepsin K (rabbit) - - - IC50 0.2nM 1nM - - - 体外研究 在体外,Odanacatib作用于组织...
n. 半胱 近义、反义、联想词 近义词n. amino acid, aminoalkanoic acid 联想词 glutathione胱;tyrosine酪;glutamate【生化】盐,酯;amino基的;protease蛋白酶;peptide;residues剩余物;enzyme酶;ligand配合基;folate叶;extracellular细胞外的; 英语例句库 1.Inhibits also some other serine and cysteine proteases lik...
A series of new dipeptidyl alpha-keto amides of the general structure R1-L-Leu-D,L-AA-CONH-R2 were synthesized and evaluated as inhibitors for the cysteine proteases calpain I, calpain II, and cathepsin B. They combine 10 different N-protecting groups (R1), 3 amino acids residues in P1...