CYP3A4*16 Reference Standard询价 产品描述 产品数据库 CBPA0098 Format Genomic DNA Description CYP3A4 (Cytochrome P450 Family 3 Subfamily A Member 4) is a Protein Coding gene. Diseases associated with CYP3A4 include Vitamin D-Dependent Rickets, Type 3 and Acetaminophen Metabolism. ...
CYP3A4, the major form of cytochrome P450 (P450) expressed in the adult human liver, is involved in the metabolism of approximately 50% of commonly prescribed drugs. Several genetic polymorphisms in CYP3A4 are known to affect its catalytic activity and to contribute in part to interindividual ...
结果:金银花提取物、绿原酸、芦丁对该酶有抑制作用,IC50值分别为2.13mg/mL、28.8μmol/L和17.6μmol/L,且金银花提取物和绿原酸对该酶的抑制作用不可逆,咖啡酸的抑制作用很弱,几乎不会导致药物相互作用。结论:金银花可能影响联合使用的CYP3A4的底物药物的代谢。
百度试题 题目葡萄柚当中含有的呋喃香豆素类化合物,可以()肠道中药物代谢酶 CYP3A4 的活性,从而减少依赖这个酶代谢的药物在肠道内的分解,()药物的吸收,导致血液中的药物浓度() 相关知识点: 试题来源: 解析 抑制;增加;升高 反馈 收藏
葡萄柚汁为肝药酶CYP3A4中效抑制剂,可受其可影响使代谢抑制和出现肌肉毒性的药品是()。A.辛伐他汀B.氯吡格雷C.苯巴比妥D.尼尔雌醇的答案是什么.用刷刷题APP,拍照搜索答疑.刷刷题(shuashuati.com)是专业的大学职业搜题找答案,刷题练习的工具.一键将文档转化为在线题库手机刷
伏立康唑通过CYP2C19、CYP2C9和CYP3A4代谢,下列可以和伏立康唑联合应用的药物是( ) A.利福平 B.卡马西平 C.奎尼丁 D.苯巴比妥 E.西咪替丁 参考答案E 解析:本题的考点是药物肝药酶代谢的相关内容。伏立康唑若与利福平(每日1次,每次600mg)合用,伏立康唑的c眦(血药峰浓度)和AUC(给药期间的血药浓度.时间...
Amlodipine metabolism in human liver microsomes and roles of CYP3A4/5 in the dihydropyridine dehydrogenation Zhu Y;Wang F;Li Q;.Amlodipine metabolism in human liver microsomes and roles of CYP3A4/5 in the dihydropyridine dehydrogenation.Drug Metab Dispos... Wang,Tang,Chen 被引量: 0发表: 0年...
Short Communication CYP3A4 * 16 and CYP3A4 * 18 Alleles Found in East Asians Exhibit Differential Catalytic Activities for Seven CYP3A4 Substrate Drugs □ ... K Maekawa,N Harakawa,T Yoshimura 被引量: 0发表: 2010年 CYP3A4*16 and CYP3A4*18 Alleles Found in East Asians Exhibit ...
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Stereoselective Metabolism of alpha-, beta-, and gamma-Hexabromocyclododecanes (HBCDs) by Human Liver Microsomes and CYP3A4中国科学院机构知识库(CAS IR GRID)以发展机构知识能力和知识管理能力为目标,快速实现对本机构知识资产的收集,长期保存,... C Erratico,X Zheng,VDE Nele,... - 《Environmental Sc...