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6. Xu, J. X.; Chen, L. B. Heteroatom Chem., 2000, 11, 158. 7. Christophe, T.; Sylviane, G. R.; Henri-Philippe, H. J. Org. Chem., 2000, 65, 6773. 8. Sekine, M.; Iimura, S.; Nakanishi, T. Tetrahedron. Lett., 1991, 32, 395...
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1,3-噻唑烷-2-硫酮在有机合成中的作用主要是通过它与羧酸或者酰卤反应生成的酰胺衍生物来表现。当1,3-噻唑烷-2-硫酮生成酰胺衍生物之后,酰基的反应活性得到活化。例如:酰胺可以被DIBAL-H 选择性还原生成相应的 醛,或者在其它酯基或者酰胺的存在下被NaBH4还原生成...
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