产品编号 T64167Cas号 1227948-82-4 别名IN-10018, BI-853520 Ifebemtinib (BI-853520) 是一种具有口服活性和强效性的粘附斑激酶 (FAK) 抑制剂 (IC50=1 nM),具有抗肿瘤活性,可抑制恶性胸膜间皮瘤中的球状体形成和原位肿瘤生长,可用于研究乳腺癌和卵巢癌。
BI-853520 CAS No. : 1227948-82-4 MCE 站:BI-853520 产品活性:BI 853520 (IN-10018) 是一种具有口服活性的粘附斑激酶 (FAK) 强效抑制剂 (重组 FAK IC50=1nM),BI 853520 表现出对癌细胞的抗增殖活性。 研究领域:Protein Tyrosine Kinase/RTK 作用靶点:FAK In Vitro: BI 853520 (0-3 μM; 2 h) ...
Product Name:BI-853520 FA(1227948-82-4 Free base) Synonyms: Ifebemtinib FA CAS: MF: MW:0 EINECS: Mol File:Mol File Browse by Nationality Suppliers >China suppliers United States (1) Member (1) All (1) Enquiry Recommend You Select Member Companies Company Name: TargetMol Chemicals In...
Phase I Study of BI 853520, an inhibitor of focal adhesion kinase, in patients with advanced or metastatic nonhematologic malignancies. Targ Oncol. 2019. https://doi.org/10.1007/s11523-018-00617-1. Article Google Scholar Doi Y, Yang JC-H, Shitara K, Naito Y, Cheng A-L, Sarashina A...
Fig. 1: BI 853520 decreases Y397-FAK phosphorylation in a dose-dependent and time-dependent manner. aTo determine the effective dose of BI 853520, 4T1, Py2T, and Py2T-LT cells were exposed to increasing concentrations of BI 853520 (0, 0.1, 0.5, 1, 5, and 10 µM for 4T1 cells...
英文名称:BI-853520 英文同义词:BI-853520;BI-853520 (BI 853520 CAS号: 分子式: 分子量:0 EINECS号: 信息错误报告 您的Email: 按国家浏览BI-853520国外供应商中国供应商 BI-853520推荐供应商 建议您优先选择企业会员,我们对企业会员产品有严格审核。
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