11.Wu F, Bhansali SG, Law WC,et al. Fluorescence imaging of the lymph node uptake of proteins in mice after subcutaneous injection: molecular weight dependence. Pharm Res. 2012 Jul;29(7):1843-53. 12.Richter WF, Bhansali SG...
②在RA中Breg出现数目和功能缺陷:研究发现,RA患者中Bregs的比例与疾病活动度呈负相关,CD24hiCD38hiBreg在RA患者中数量减少且存在功能缺陷,无法抑制Th17反应和将C D 4 + T细胞转化为调节性T细胞(regulatory T cell,Treg)[9]。此外,RA患者与健康人相比,IL-10+TIM1+ Breg细胞和IL-10+CD5+CD1dhiBreg细胞比例...
静脉输注0.9%生理盐水1 L 或10~15 ml/kg(如60 kg,600~900 ml/d静脉输注);服用口服补液盐(在开始输注AmB前60 min口服1 L;当天剩下的时间分次口服2 L,根据患者耐受性评估酌情调整),已被证明是一个实用简单的方法但更有效的替代方案,尿钠排泄量...
[4]. Meng Q, et al. Protective Effects of Alisol B 23-Acetate Via Farnesoid X Receptor-Mediated Regulation of Transporters and Enzymes in Estrogen-Induced Cholestatic Liver Injury in Mice. Pharm Res. 2015 Jun 4. 公司简介 武汉科斯坦生物科技有限公司是一家致力于前沿生物技术研发与成果转化的创新型...
DrugsStatusIndicationsR&D Company Ibrutinib launched CLL, MCL, WM, ABC-DLBCL Pharmacyclics/Johnson Acalabrutinib launched MCL AstraZeneca/Acerta Pharm BV Zanubrutinib launched CLL, MCL, FL, WM, SLL BeiGene Orelabrutinib NDA MCL, CLL, SLL, WM Avila/Celegene Tirabrutinib launched Recurrent...
Etalocib (LY293111) 是具有口服活性的白三烯 (LTB4) 受体的拮抗剂,抑制 [3H]LTB4 结合的Ki 值为 25 nM. Etalocib (LY293111) 抑制LTB4 诱导的钙动员的 lC50 值为 20 nM。Etalocib (LY293111) 可诱导凋亡。 体外研究 Etalocib (LY293111) elicits a concentration-dependent inhibition of LTB4induced CD...
Medically Reviewed bySimi Burn, PharmDon Aug 25, 2024 | Written byCourtney Zeigler, PharmD, BCPS Common Brand Name(s):Neo-Polycin Common Generic Name(s):Neosporinneomycin/polymyxin B/gramicidin ophthalmic, neomycin sulfate/polymyxin B sulfate/gramicidin D ...
Vazin A, Karimzadeh I, Zand A, Hatami-Mazinani N, Firouzabadi D. Evaluating adherence of health-care team to standard guideline of colistin use at intensive care units of a referral hospital in Shiraz, southwest of Iran. Adv Pharm Bull. 2017;7(3):391–7. https://doi.org/10.15171/ap...
Medically Reviewed by Morgan Corbin, CPP, PharmD, BCOP on Jun 25, 2024 | Written by Dena Westphalen, PharmD Common Brand Name(s): Retevmo Common Generic Name(s): selpercatinib Pronunciation: reh-TEHV-moh, SEL-per-KA-tih-nib Drug Classes: antineoplastic, kinase inhibitor Availability: pre...
cAmB以两性霉素B脱氧胆酸盐(D-AmB)为经典制剂,D-AmB进入血液后,AMB分子与脱氧胆酸盐分离,以游离形式存在并发挥作用,AMB通过与真菌细胞膜上的麦角固醇结合,在细胞膜上形成管状离子通道,使得电解质等胞内物质外流从而导致真菌细胞死亡[4]。 研究发现...