AR-C118925 is a potent and selective non-nucleotide antagonist blocking P2Y2 receptors with a pA2 value of 7.8 (Kemp et al., 2004; Kindon et al., 2017; Rafehi et al., 2017a, 2017c). The P2Y2 receptor is widely expressed (von Kügelgen and Wetter, 2000; Abbracchio et al., ...
ins were not inhibited by the P2Y2R antagonist AR-C118925, and the receptor desensitization profile suggested the involvement of FPR2 rather than P2Y2... M Gabl,R Holdfeldt,M Winther,... - Biochimica et Biophysica Acta (BBA) - Molecular Cell Research 被引量: 9发表: 2016年 Discovery ...