The results obtained indicate that steric interactions are crucial for antimycobacterial activity, while hydrogen bond donor groups participate negligibly in activity. The derived 3D㏎SAR models showed acceptable r (0.91) and q (0.91) with a root mean squared error (RMSE) of 0.08. The models ...
1) antimycobacterial activity 抗快速增殖分枝杆菌活性 1. Synthesis andantimycobacterial activityof 3-substituted benzoyl-4H-chromen-4-ones 3-取代苯甲酰基-4H-色烯-4-酮的合成及其抗快速增殖分枝杆菌活性研究 更多例句>> 2) activity against mycobacteria ...
Antimycobacterial activity of some Brazilian indigenous medicinal drinks. J Basic Appl Pharm Sci 2007;28:165‑9.Oliveira DG, Prince KA, Higuchi CT, Santos ACB, Lopes LMX, Simões MJS, et al. Antimycobacterial activity of some Brazilian indigenous medicinal drinks. J Basic Appl Pharm Sci. ...
antimycobacterial activityMICtoxicity (IC50A series of 7-O-alkoxy-4-methylumbelliferone derivatives were prepared using a convenient one step synthesis. Additionally the bromo- and azido derivatives 7-O-(4-bromobutoxy)-, 7-O-(6-bromohexyloxy)- and 7-O-(6-azidohexyloxy)-4-methylumbelliferone ...
all commonly used in the treatment of microbial infections [24]. Even though there are no approved anti-TB drugs of fungal origin to date, there are numerous fungal-derived compounds which have been previously shown to possess strong natural antimycobacterial activity which is comparable to that of...
Synthesis and Preliminary In Vitro Evaluation of Antimycobacterial Activity of New Pyrrolo[1,2- a ]quinoxaline-carboxylic Acid Hydrazide Derivatives[J] . Jean Guillon,Robert C. Reynolds,Jean-Michel Leger,Marie-Aude Guie,Stephane Massip,Patrick Dallemagne,Christian Jarry.Journal of Enzyme Inhibition ...
Evaluates the in vitro antimycobacterial activity of BAY 12-8039, a methoxyfluoroquinolone. Materials and methods; Results and discussion.doi:10.2165/00003495-199958002-00139Dr Hajime SaitoSpringer International PublishingDrugsSaito H. Comparative antimycobacterial activity of BAY 12- 8039 and gatifloxacin. ...
Synthesis and antimycobacterial activity of some coupling products from 4-aminobenzoic acid hydrazones. European Journal of Medicinal Chemistry . 1999; 34 (12):1093–1100.Kucukguzela, S.G.; Rollas, S.; Kucukguzel, I.; Kiraz, M. Synthesis and antimycobacterial activity of some coupling products ...
Thus, as a main goal of this study, rifampicin nanoparticles were surface functionalized with a tuftsin-modifed peptide to selectively recognize receptors located on infected alveolar macrophages, enhancing nanoparticles uptake by these cells and improving antimycobacterial activity. A tuftsin-based ...
Antimycobacterial Activity and Alkaloid Prospection of Psychotria Species (Rubiaceae) from the Brazilian Atlantic Rainforest.Antimycobacterial Activity and Alkaloid Prospection of Psychotria Species (Rubiaceae) from the Brazilian Atlantic Rainforest.doi:10.1055/s-0030-1250656alkaloids...