Examples of such acids are 6-(5-benzoylvaleramido), 6-(3-benzoylpropionamido), 6-[3-(2,4,6-trimethoxy - benzoyl) propionamido], 6 - [4 - (2, 4 - dichloro - benzoyl) butyramido], 6 - [3 - (2, 4 - dihydroxy - benzoyl) propionamido], 6 - [3 - (3 - diethyl - ...
2024 The researchers speculate that the metals could be finding their way into tampon products via contaminated cotton, or that some metals may be intentionally added during manufacturing to whiten materials or as antibacterial agents, for example. Tanyel Mustafa, refinery29.com, 12 July 2024 The ...
organic antibacterial agents, and hydrogel-based agents exhibit good antibacterial activity, providing the new strategies for the treatment of bacterial diseases [13,14,15]. Among them, hydrogel, as a kind of good antibacterial materials, can be used with a variety of antibacterial agents to achiev...
Antibacterial agents United States Patent 4132712 Abstract: Compounds of the formula ##STR1## wherein CO2R is an ester group, are useful for their β-lactamase inhibitory activity. Inventors: Howarth, Thomas T. (Ewhurst, GB2) Stirling, Irene (Worcester Park, GB2)...
This Chapter covers the role of chirality in the antibacterial activity and the consequence of this chirality in terms of chemical synthesis by showing characteristic examples within the main classes of antibacterial agents, including β-lactams, β-lactamase inhibitors, glycopeptides, fosfomycin, ...
et al. Discovery of a novel and potent class of FabI-directed antibacterial agents. Antimicrob. Agents Chemother. 46, 3118–3124 (2002). References 13 and 14 describe the development of antibacterial compounds from enzyme inhibitors that had little initial antibacterial activity. CAS PubMed PubMed...
The scope of our current work is based on the hypothesis that the different physicochemical properties of antibacterial agents may also be related to the nature and type of their molecular targets responsible for drug efficacy. Here we focus on differences in the surface properties of the binding ...
The cytotoxicity against HEKa cells provides useful toxicology information for the development of safe, topically-applied antibacterial agents [65,66]. In this research program, HEKa cells were differentiated to a stratified squamous epithelium via an air–liquid interface; this type of epithelium can ...
Cell wall active agents are believed to increase damaged or mis-folded proteins and result in induction of genes involved in protein turnover such as chaperones and proteases [[Muthaiyan et al., Antimicrob Agents Chemother 52:980-990 (2008); Utaida et al., Microbiology 149:2719-2732 (2003)...
Antifungal activity of liriodenine on agents of systemic mycoses, with emphasis on the genus Paracoccidioides. J. Venom. Anim. Toxins Incl. Trop. Dis. 2020, 26, e20200023. [Google Scholar] [CrossRef] Ashraf, S.M.; Mahanty, S.; Rathinasamy, K. Securinine induces mitotic block in ...