表2 本发明化合物α-葡萄糖苷酶活性研究(x士S,n=2) α-淀粉酶活性研究表明,20(R)-原人参三醇(PPT)等系列人参皂苷对α-淀粉酶具有极强的抑制活性,其中25-OCH3-PPT和25-OH-PPT对α-葡萄糖苷酶抑制活性强于阳性对照药阿卡波糖(acarbose)。几种衍生物中25-OH-PPT对α-葡萄糖苷酶抑制作用最强,其抑制率达到...
Of the four test compounds, 25-OCH3-PPD was most potent. It decreased survival, inhibited proliferation, induced apoptosis, and led to G1 cell cycle arrest in both cell lines. It also decreased the levels of proteins associated with cell proliferation (MDM2, E2F1, cyclin D1, and cdks 2 ...
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