Design and synthesis of (4E)-4-(4-substitutedbenzylideneamino)-3- substituted-2,3-dihydro-2-thioxothiazole-5-carbonitrile as novel A2A receptor antagonistsA2AR antagonistHaloperidol 2-ThioxothiazoleRadioligand-binding assay cAMP assayNovel 2-thioxothiazole derivatives (6-19) as potential adenosine A ...
The present invention relates to novel synthesis of 4E)-4-(4-substituted benzy1ideneamino)- 2,3-dihydro-3-substituted -2-thioxothiazole-Scarbonitriles of general formula 2 wherein R and R1 are selected from a group consisting of wherein R is selected from a group consisting of hydrogen, ...
Synthesis of Novel Biologically Important 5-Amino-2-Oxo-7-Aryl-3,7-Dihydro-2H-Pyrano[2,3-d]Thiazole-6-Carbonitriles in Trifluoroethanol (TFE) under Ultrasound Irradiation Condition and Their Antimicrobial ActivityMulticomponent reactions2H-pyrano[23-d]thiazole-6-carbonitriles...