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将颈、胸、腰椎和颅骨皮质骨中PET/CT引导VOI分别定义用于骨髓或骨骼评估。注射后1h, 18 F-GLN在小鼠骨髓摄取相对较高,高达(9.5±1.3)%ID/g,是 18 F-FLT的2.1倍。化疗药物明显抑制了骨髓 18 F-GLN的摄取。 18 F-GLN骨髓摄取的减少与白细胞减少(骨髓抑制)一致。对于人体 18 F-GLN PET显像,静脉注射后1h,...
We report the preparation of a novel glutamine derivative, (2S,4S)-2,5-diamino-4-(4-(2-fluoroethoxy)benzyl)-5-oxopentanoic acid, (2S, 4S)4-[18F]FEBGln ([18F]4), through efficient organic and radiosyntheses. In vitro assays of [18F]4 using MCF-7 cells showed that it entered ...
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Structure of 1 (BAY 85-8050), 2 ([18F](2S, 4R)4F-GLN), 3 (BAY 94-9392), and 4 ([18F]FPMET).Hu, KongzhenDu, KanTang, GanghuaYao, ShaoboWang, HongliangLiang, XiangYao, BaoguoHuang, TingtingZang, Linquan