1,3-Diazolyl-2-propanol derivatives of the formula wherein X and Y are N or CH, R1 is phenyl, heterocyclyl, heterocyclyl-alkyl, -alkenyl or -alkynyl, optionally substituted, R2 and R3 are hydrogen or alkyl, and R4 and R5 are hydrogen, amino, alkoxyalkyl, aminoalkyl, alkylaminoalkyl,...
近日,来自波兰卢布林医科大学药学院生物与遗传学系的研究者们在J Adv Res杂志上发表了题为“Synthesis and anthelmintic activity of novel thiosemicarbazide and 1,2,4-triazole derivatives: In vitro, in vivo, and in silico study”的文章,该研究表明在体外、体内和硅研究中,化合物II-1可以被描述为HIT,未来...
近日,来自波兰卢布林医科大学药学院生物与遗传学系的研究者们在J Adv Res杂志上发表了题为“Synthesis and anthelmintic activity of novel thiosemicarbazide and 1,2,4-triazole derivatives: In vitro, in vivo, and in silico study”的文章,该研究表明在体外、体内和硅研究中,化合物II-1可以被描述为HIT,未来...
OF THE DISCLOSURE:\nThe invention is concerned with new derivatives\nof 1, 2, 4-triazole having the general formula:\n(I)wherein:\nX = O or S;\nR3 = H, alkyl containing from 1 to 5 carbon atoms,\nC6H5, benzyl, alkenyl containing from 2 to 6 carbon\natoms, or alkynyl containing ...
Plant protecting agents based on 1,2,4 - triazole derivatives as well as 1,2,4-triazole derivatives not available for EP017456of corresponding document:The invention relates to plant protection agents which contain a triazole compound of the formula I (I) in which Z denotes halogen, nitro, ...
1,2,4-Triazole derivatives possess a varied of pharmacological properties such as anti-tubercular, anti-fungal, anti-tumor and anti-bacterial activities due to 1,2,4-triazole moiety can exert various non-covalent interactions that are able to improve the solubility and the ability of binding to...
1,2,4-三唑类衍生物 例句>> 3) 3-methyl-4-amino-5-mercapto-1,2,4-triazole derivatives 3-甲基-4-氨基-5-巯基-1,2,4-三唑衍生物 1. Synthesis and antifungal activity of 3-methyl-4-amino-5-mercapto-1,2,4-triazole derivatives; 3-甲基-4-氨基-5-巯基-1,2,4-三唑衍生物的合成及抗...
近日,来自波兰卢布林医科大学药学院生物与遗传学系的研究者们在J Adv Res杂志上发表了题为“Synthesis and anthelmintic activity of novel thiosemicarbazide and 1,2,4-triazole derivatives: In vitro, in vivo, and in silico study”的文章,该研究表明在体外、体内和硅研究中,化合物II-1可以被描述为HIT,未来...
1,2,4-三唑衍生物 1. To explore the synthesis and photophysical properties of 1,2,4-triazole derivatives,4-amino-3,5-bis(o-hydroxyphenyl)-1,2,4-triazole was synthesized by improved methods of dihydrazide cyclization. 为探索1,2,4-三唑衍生物的合成及光物理性能,通过改进的双酰肼环化法合成了...
Novel vasopressin V2 receptor-selective antagonists, pyrrolo[2,1-a]quinoxaline and pyrrolo[2,1-c][1,4]benzodiazepine derivatives Synthesis and structure-activity relationships (SAR) of a novel series of vasopressin V(1b) antagonists are described. 2-(6-Aminomethylaryl-2-aryl-4-oxo-quinazolin-3...