properties and α-glucosidase inhibitory activity of WAFP were in- vestigated. 2. Materials and methods 2.1. Materials and chemicals Fresh wax apple (Syzygium samarangense Merr. & Perry) fruits were purchased from Sanya (Hainan Province, China). Before the extraction, the fruits were washed, pe...
Synthesis and α-glucosidase inhibitory activity of N-(1,5-diaryl-3-pentone-1-yl)-4-aminobenzoic acid N-(1,5-二芳基-3-戊酮-1-基)-4-氨基苯甲酸的合成与α-葡糖苷酶抑制活性初步研究 3. The seminal plasma components of free L-carnitine,α-glucosidase,fructose and acid phosphatase were det...
The work includes α-glucosidase inhibitory activity of sericin with special focus on its interaction with the enzyme, study of thermodynamic parameters and molecular modeling. Sericin inhibited α-glucosidase (IC50=2.9 μM) in a noncompetitive fashion (Ki=1.0 μM); it binds to the enzyme at a...
Piper trioicum, Hypoglycemic Activity, Alpha-Glucosidase Inhibition. Therapeutic Drug Monitoring Abstract Alpha glucosidasein vitroinhibitory activity and hypoglycemic effect by oral administration in rats ofPiper trioicumethanol extracts have been investigated.Piper trioicumextract showedin vitroinhibitory activ...
aThe α-glucosidase inhibitory activity of the OTPS was determined according to the method described by Apostolidis and Lee with a slight modification. OTPS的α葡糖苷酶禁止活动根据Apostolidis和李描述的方法是坚定的以轻微的修改。[translate]
In present study synthesized thirty quinazolinone compounds (PM1-PM30) were screened for their inhibitory effect on alpha amylase and alpha glucosidase enzymes. All synthesized compounds PM1 to PM 30, possess good inhibitory activity similar to that of approved drug Acarbose. Compounds PM20 PM7, PM...
The brown seaweed Sargassum hemiphyllum exhibits α-amylase and α-glucosidase inhibitory activity and enhances insulin release in vitro The brown seaweed sargassum hemiphyllum exhibits alpha-amylase and alpha-glucosidase inhibitory activity and enhances insulin release in vitro. Cytotechnology ... Pai-...
The secretion of gastric inhibitory polypeptide (GIP) may be reduced whereas secretion of glucagon-like peptide-1 (7-36 amide) (GLP-1) is increased.19 When used as monotherapy in patients complying with dietary advice, an α-alpha-glucosidase inhibitor can be expected to reduce peak ...
Salazinic Acid-Derived Depsidones and Diphenylethers with α-Glucosidase Inhibitory Activity from the Lichen Parmotrema dilatatum Three new depsidones, parmosidones F – G (1 – 2), and 8′-O-methylsalazinic acid (3), and 3 new diphenylethers, parmetherines A – C (4 – 6), together...
The ethyl acetate (EtOAc) fraction exhibited the most significant inhibitory activity. Eight pure compounds, apigenin, apigenin-7-O-β-D- glucoside, kaempferol, hyperin, naringenin, quercetin, luteolin, and kaempferol-7-O-β-D- glucoside, were isolated (using enzyme assay-guide fractionation ...